SCHEMBL10187477

SCHEMBL10187477

Cc1cccc(-c2cnc([C@]3(C)CC(=O)N(C)C(=N)N3)s2)c1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 3/20 0.38
HSD17B2 P37059 3/20 0.38
BACE1 P56817 5/20 0.37
BACE2 Q9Y5Z0 2/20 0.37
HDAC1 Q13547 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
PGR P06401 1/20 0.32
GRIN1 Q05586 1/20 0.32
GRIN2B Q13224 1/20 0.32
KDR P35968 1/20 0.31
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30
SYK P43405 1/20 0.30
ADORA3 P0DMS8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2962946 0.89 BACE1 (0.36) BACE1BACE2SLC6A2SLC6A4SLC6A3
SCHEMBL2956532 0.89 BACE1 (0.36) BACE1BACE2HDAC1HDAC6PGR
SCHEMBL13081360 0.89 BACE1 (0.36) BACE1BACE2
SCHEMBL2962943 0.89 BACE1 (0.36) BACE1BACE2SLC6A2SLC6A4SLC6A3
SCHEMBL2956526 0.89 BACE1 (0.36) BACE1BACE2HDAC1HDAC6PGR
SCHEMBL14106041 0.89 HSD17B1 (0.42) HSD17B1HSD17B2BACE1BACE2
SCHEMBL15291996 0.88 BACE1 (0.40) BACE1BACE2
SCHEMBL4557056 0.87 BACE1 (0.35) BACE1BACE2
SCHEMBL7566391 0.86 BACE1 (0.49) BACE1BACE2PGR
SCHEMBL7605403 0.85 WRN (0.42) BACE1BACE2GRIN1GRIN2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120232064-A1 ASPARTYL PROTEASE INHIBITORS SCHERING CORPORATION (US) 2012-09-13 US disclosed
US-8168641-B2 Aspartyl protease inhibitors SCHERING CORPORATION (US) 2012-05-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120232064-A1 ASPARTYL PROTEASE INHIBITORS CHRM1, CHRM2, BACE1 HSD17B1 1676/4885HSD17B2 2823/4885BACE1 3/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.