SCHEMBL10187496

SCHEMBL10187496

O=c1[nH]c(-c2cccc(S)c2)no1

nearest known ligand 0.47

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.44
PARP1 P09874 1/20 0.42
PDE5A O76074 1/20 0.41
PDE1A P54750 1/20 0.41
PDE1B Q01064 1/20 0.41
PDE4D Q08499 1/20 0.41
PDE7A Q13946 1/20 0.41
PDE1C Q14123 1/20 0.41
PDE3A Q14432 1/20 0.41
RARB P10826 2/20 0.41
ADH5 P11766 1/20 0.40
KMO O15229 1/20 0.40
IDO1 P14902 1/20 0.39
RARG P13631 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2645918 0.81 ALDH1A1 (0.45) ALDH1A1PARP1PDE5APDE1APDE1B
SCHEMBL15059204 0.80 GRIK1 (0.46) ALDH1A1PARP1PDE5APDE1APDE1B
SCHEMBL4504146 0.80 ALDH1A1 (0.46) ALDH1A1PARP1PDE5APDE1APDE1B
SCHEMBL18603181 0.80 NOTUM (0.50) ALDH1A1PDE5APDE1APDE1BPDE4D
SCHEMBL2645921 0.80 PARP1 (0.45) ALDH1A1PARP1PDE5APDE1APDE1B
SCHEMBL8295573 0.80 NOTUM (0.50) ALDH1A1PDE5APDE1APDE1BPDE4D
SCHEMBL18603164 0.80 NOTUM (0.50) ALDH1A1PARP1PDE5APDE1APDE1B
Hydrochloric Acid SCHEMBL4512162 0.79 ALDH1A1 (0.45) ALDH1A1PARP1PDE5APDE1APDE1B
SCHEMBL3743779 0.78 ALDH1A1 (0.56) ALDH1A1PARP1RARBADH5RARG
SCHEMBL481019 0.78 BRD4 (0.49) ALDH1A1PARP1PDE5APDE1APDE1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012058203-A1 DIAZENIUMDIOLATE HETEROCYCLIC DERIVATIVES MERCK SHARP & DOHME CORP. (US) 2012-05-03 WO disclosed