SCHEMBL10194085

SCHEMBL10194085

CO/C(N)=N/Cc1cccc(NC(=O)c2ccc(N)cn2)c1

nearest known ligand 0.50

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
ACKR3 P25106 1/20 0.50
BACE1 P56817 10/20 0.48
ALDH1A1 P00352 2/20 0.43
POLB P06746 1/20 0.43
MEN1 O00255 1/20 0.43
LMNA P02545 1/20 0.43
KMT2A Q03164 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
SIRT2 Q8IXJ6 6/20 0.42
SIRT1 Q96EB6 6/20 0.42
SIRT3 Q9NTG7 6/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10195043 0.91 BACE1 (0.49) ACKR3BACE1ALDH1A1POLBMEN1
SCHEMBL10194903 0.89 BACE1 (0.45) ACKR3BACE1ALDH1A1POLBMEN1
SCHEMBL10193692 0.86 ACKR3 (0.44) ACKR3BACE1ALDH1A1POLBMEN1
SCHEMBL10192948 0.85 BACE1 (0.51) BACE1
SCHEMBL10193690 0.85 ACKR3 (0.44) ACKR3BACE1ALDH1A1POLBMEN1
SCHEMBL10194912 0.81 PRSS1 (0.46) ACKR3BACE1ALDH1A1POLBMEN1
SCHEMBL10193576 0.81 NPC1 (0.43) BACE1SMN1; SMN2
SCHEMBL10193143 0.78 BACE1 (0.47) BACE1
SCHEMBL10193709 0.77 SMN1; SMN2 (0.42) ACKR3BACE1ALDH1A1POLBMEN1
SCHEMBL10194093 0.77 BACE1 (0.42) ACKR3BACE1ALDH1A1POLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2415756-A1 ISOTHIOUREA DERIVATIVES OR ISOUREA DERIVATIVES HAVING BACE1 INHIBITORY ACTIVITY Shionogi&Co., Ltd. (JP) 2012-02-08 EP disclosed