SCHEMBL10200243

SCHEMBL10200243

C#Cc1ccc2c(ccc3nc([C@@H]4CCCN4)[nH]c32)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN10A Q9Y5Y9 1/20 0.45
CDC7 O00311 13/20 0.36
CCNE1 P24864 9/20 0.36
CDK2 P24941 9/20 0.36
ROCK1 Q13464 9/20 0.36
DBF4 Q9UBU7 9/20 0.36
PIM1 P11309 4/20 0.35
CSNK2B P67870 4/20 0.35
CSNK2A1 P68400 4/20 0.35
DYRK1A Q13627 3/20 0.35
CIT O14578 1/20 0.35
CYP1A2 P05177 1/20 0.35
CSNK2A2 P19784 1/20 0.35
GSK3B P49841 1/20 0.35
CSNK2A3 Q8NEV1 1/20 0.35
TAOK3 Q9H2K8 1/20 0.35
PARP1 P09874 3/20 0.34
TYMS P04818 1/20 0.34
CCNC P24863 2/20 0.33
CDK8 P49336 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10201776 0.85 SCN10A (0.53) SCN10ACDC7CCNE1CDK2ROCK1
SCHEMBL14758479 0.82 CDC7 (0.48) SCN10ACDC7CCNE1CDK2ROCK1
SCHEMBL12373613 0.81 TYMS (0.33) TYMS
SCHEMBL10236922 0.80 SCN10A (0.38) SCN10ACDC7CCNE1CDK2ROCK1
SCHEMBL19488489 0.80 CDC7 (0.38) SCN10ACDC7CCNE1CDK2ROCK1
SCHEMBL12798759 0.79 SCN10A (0.52) SCN10ACDC7CCNE1CDK2ROCK1
SCHEMBL12404403 0.79 SCN10A (0.56) SCN10ACDC7CCNE1CDK2ROCK1
SCHEMBL10201770 0.79 SCN10A (0.41) SCN10ACDC7CCNE1CDK2ROCK1
SCHEMBL13561572 0.78 SCN10A (0.44) SCN10ACDC7CCNE1CDK2ROCK1
SCHEMBL10200241 0.78 TYMS (0.33) TYMS

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012018325-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-09 WO disclosed