SCHEMBL10200595

SCHEMBL10200595

COCn1cc(N)cn1

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1663037 0.80 MEN1 (0.45)
SCHEMBL17508623 0.80 MEN1 (0.42)
SCHEMBL31599691 0.77 MEN1 (0.40)
SCHEMBL14764041 0.77 MEN1 (0.43)
SCHEMBL10174579 0.77
SCHEMBL22980532 0.76 L3MBTL1 (0.44)
SCHEMBL5928297 0.76 MEN1 (0.39)
SCHEMBL19011387 0.76 MEN1 (0.42)
SCHEMBL174144 0.76
SCHEMBL31579078 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12459925-B2 Sulphonyl urea derivatives as NLRP3 inflammasome modulators NodThera Limited (GB) 2025-11-04 US disclosed
US-20250333424-A1 ANTIVIRAL COMPOUNDS GILEAD SCIENCES, INC. 2025-10-30 US disclosed
EP-3728238-B1 SULPHONYL UREA DERIVATIVES AS NLRP3 INFLAMMASOME MODULATORS NODTHERA LTD (GB) 2025-06-18 EP disclosed
CN-119241539-A Pyrazolo piperidine (ketone) -containing derivative, and preparation method and application thereof 沈阳药科大学 2025-01-03 CN disclosed
US-20240368129-A1 SULPHONYL UREA DERIVATIVES AS NLRP3 INFLAMMASOME MODULATORS NodThera Limited (GB) 2024-11-07 US disclosed
CN-116396205-B N-aryl indole derivative and preparation method and application thereof 沈阳药科大学 2024-10-01 CN disclosed
US-12012397-B2 Sulphonyl urea derivatives as NLRP3 inflammasome modulators NodThera Limited (GB) 2024-06-18 US disclosed
CN-116396205-A N-aryl indole derivative and preparation method and application thereof 沈阳药科大学 2023-07-07 CN disclosed
US-20230145050-A1 SULPHONYL UREA DERIVATIVES AS NLRP3 INFLAMMASOME MODULATORS NodThera Limited (GB) 2023-05-11 US disclosed
US-11518757-B2 Sulphonyl urea derivatives as NLRP3 inflammasome modulators NodThera Limited (GB) 2022-12-06 US disclosed
CN-111954670-A Sulfonylurea derivatives as NLRP3 inflammasome modulators 诺瑟拉有限公司 2020-11-17 CN disclosed
EP-3728238-A1 SULPHONYL UREA DERIVATIVES AS NLRP3 INFLAMMASOME MODULATORS Nodthera Limited (GB) 2020-10-28 EP disclosed
US-8569336-B2 Compounds for the treatment of inflammatory disorders TONG LING (US) 2013-10-29 US disclosed
US-8569336-B2 Compounds for the treatment of inflammatory disorders TONG LING (US) 2013-10-29 US disclosed
US-8450355-B2 Compounds for the treatment of inflammatory diseases MERCK SHARP & DOHME CORP. (US) 2013-05-28 US disclosed
US-8450355-B2 Compounds for the treatment of inflammatory diseases MERCK SHARP & DOHME CORP. (US) 2013-05-28 US disclosed
US-20120015926-A1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS TONG LING (US) 2012-01-19 US disclosed
US-20120015926-A1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISORDERS TONG LING (US) 2012-01-19 US disclosed
US-20110288077-A1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISEASES SCHERING CORPORATION (US) 2011-11-24 US disclosed
US-20110288077-A1 COMPOUNDS FOR THE TREATMENT OF INFLAMMATORY DISEASES SCHERING CORPORATION (US) 2011-11-24 US disclosed