SCHEMBL10201478

SCHEMBL10201478

O=C(OCc1ccccc1)N1C2C[C@@H]2C[C@H]1c1nc2c([nH]1)-c1ccc(Br)cc1CC2

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 1/20 0.36
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
L3MBTL1 Q9Y468 1/20 0.34
DHFR P00374 1/20 0.34
KDR P35968 1/20 0.34
AGTR2 P50052 4/20 0.33
AAK1 Q2M2I8 1/20 0.33
PARP1 P09874 1/20 0.33
KCNK3 O14649 1/20 0.33
KCNK9 Q9NPC2 1/20 0.33
TYMS P04818 1/20 0.33
GRIN2B Q13224 1/20 0.33
PSEN1 P49768 1/20 0.32
PSEN2 P49810 1/20 0.32
APH1B Q8WW43 1/20 0.32
NCSTN Q92542 1/20 0.32
APH1A Q96BI3 1/20 0.32
PSENEN Q9NZ42 1/20 0.32
SRD5A1 P18405 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3425525 1.00 HTR2C (0.36) HTR2CNPC1RAB9AL3MBTL1DHFR
SCHEMBL10232542 1.00 HTR2C (0.36) HTR2CNPC1RAB9AL3MBTL1DHFR
SCHEMBL13747270 1.00 HTR2C (0.36) HTR2CNPC1RAB9AL3MBTL1DHFR
SCHEMBL10233657 0.86 HTR2C (0.43) HTR2CNPC1RAB9AL3MBTL1DHFR
SCHEMBL2066099 0.85 TYMS (0.39) TYMSSRD5A1SRD5A2
SCHEMBL19488761 0.83 HTR2C (0.37) HTR2CNPC1RAB9AL3MBTL1DHFR
SCHEMBL2065597 0.83 TYMS (0.35) TYMSSRD5A1SRD5A2
SCHEMBL2065596 0.83 TYMS (0.35) TYMSSRD5A1SRD5A2
SCHEMBL13746544 0.83 TYMS (0.35) TYMSSRD5A1SRD5A2
SCHEMBL883262 0.83 TYMS (0.35) TYMSSRD5A1SRD5A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012018325-A1 HEPATITIS C VIRUS INHIBITORS BRISTOL-MYERS SQUIBB COMPANY (US) 2012-02-09 WO disclosed