SCHEMBL10205608

SCHEMBL10205608

Cc1nc(Nc2cccc3ccccc23)sc1CCON(O)O

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 8/20 0.45
MAPT P10636 5/20 0.44
KDM4E B2RXH2 3/20 0.44
ALDH1A1 P00352 3/20 0.44
GAA P10253 2/20 0.44
MEN1 O00255 3/20 0.43
KMT2A Q03164 3/20 0.43
POLB P06746 2/20 0.43
PTGDR2 Q9Y5Y4 1/20 0.43
NPC1 O15118 2/20 0.42
RAB9A P51151 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
HPGD P15428 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
CDC25A P30304 1/20 0.39
CDC25B P30305 1/20 0.39
CDC25C P30307 1/20 0.39
CASP3 P42574 1/20 0.39
SENP7 Q9BQF6 1/20 0.39
SENP6 Q9GZR1 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL279243 0.86 PTGDR2 (0.43) MAPTKDM4EALDH1A1GAAMEN1
SCHEMBL6273265 0.84 CCR4 (0.50) CCR4MAPTKDM4EALDH1A1GAA
SCHEMBL280339 0.83 GAA (0.55) MAPTKDM4EALDH1A1GAAMEN1
SCHEMBL6270866 0.83 CCR4 (0.44) CCR4MAPTKDM4EALDH1A1GAA
SCHEMBL263590 0.81 CCR4 (0.43) CCR4MAPTKDM4EALDH1A1GAA
SCHEMBL279897 0.79 HTR2C (0.50) KDM4EALDH1A1HPGD
SCHEMBL280460 0.77 GAA (0.40) MAPTKDM4EALDH1A1GAAMEN1
SCHEMBL280302 0.77 ITGB3 (0.32) ALDH1A1
SCHEMBL12646824 0.76 PTGDR2 (0.45) MAPTKDM4EALDH1A1GAAMEN1
SCHEMBL280485 0.74 DHODH (0.40) MAPTKDM4EALDH1A1GAAPTGDR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8134010-B2 4-[4-Methyl-5-(2-nitrooxy-ethyl)-thiazol-2-yl]-phenylamine; N-{4-[4-Methyl-5-(2-nitrooxy-ethyl)-thiazol-2-yl]-phenyl}-acetamide; or4-Methyl-5-(2-nitrooxy-ethyl)-2-(4-nitro-phenyl)-thiazole; cardiovascular, gastrointestinal, inflammatory, respiratory disease RENOPHARM LTD. (IL) 2012-03-13 US disclosed