SCHEMBL10205609

SCHEMBL10205609

CCOC(=O)c1cc(C)c(OC(=O)CCCc2ccc(NC(=O)c3ccc(C)nc3-c3ccc(C(F)(F)F)cc3)c(C(=O)N(C)C)c2)c(C)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NTRK1 P04629 1/20 0.42
NTRK2 Q16620 1/20 0.42
PLK1 P53350 1/20 0.36
NFKB1 P19838 2/20 0.34
ATF1 P18846 1/20 0.34
MAOB P27338 1/20 0.34
MTTP P55157 1/20 0.33
PPARG P37231 3/20 0.33
PPARA Q07869 2/20 0.33
KDM4E B2RXH2 3/20 0.32
MEN1 O00255 2/20 0.32
MAPT P10636 2/20 0.32
KMT2A Q03164 2/20 0.32
HSP90AA1 P07900 1/20 0.32
CRHBP P24387 1/20 0.32
CRHR2 Q13324 1/20 0.32
CETP P11597 1/20 0.32
PTGES O14684 1/20 0.32
HTT P42858 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL402751 0.96 NTRK1 (0.40) NTRK1NTRK2PLK1NFKB1ATF1
SCHEMBL401200 0.95 NTRK1 (0.40) NTRK1NTRK2PLK1NFKB1ATF1
SCHEMBL402835 0.95 NTRK1 (0.40) NTRK1NTRK2PLK1NFKB1ATF1
SCHEMBL403797 0.95 NTRK1 (0.40) NTRK1NTRK2PLK1NFKB1ATF1
SCHEMBL403346 0.95 NTRK1 (0.42) NTRK1NTRK2PLK1MTTPPPARG
SCHEMBL402008 0.93 NTRK1 (0.41) NTRK1NTRK2PLK1NFKB1ATF1
SCHEMBL5316686 0.93 NTRK1 (0.42) NTRK1NTRK2PLK1MTTPPPARG
SCHEMBL401854 0.92 NTRK1 (0.40) NTRK1NTRK2PLK1NFKB1ATF1
SCHEMBL402750 0.91 NTRK1 (0.40) NTRK1NTRK2PLK1MTTPPPARG
SCHEMBL400959 0.91 NTRK1 (0.40) NTRK1NTRK2PLK1MTTPPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed
US-8101774-B2 Ester derivatives and medicinal use thereof JAPAN TOBACCO INC. (JP) 2012-01-24 US disclosed