SCHEMBL10214943

SCHEMBL10214943

C=C1NC(=O)CCC1n1c(C)nc2cccc(CN)c2c1=O

nearest known ligand 0.60

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 18/20 0.60
CRBN Q96SW2 18/20 0.60
IKZF3 Q9UKT9 3/20 0.60
TNF P01375 2/20 0.60
IL1B P01584 2/20 0.60
GAA P10253 1/20 0.34
ALOX15 P16050 1/20 0.34
TBXA2R P21731 1/20 0.32
IKZF1 Q13422 1/20 0.32
KDM4E B2RXH2 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18900402 0.92 DDB1 (0.60) DDB1CRBNIKZF3TNFIL1B
SCHEMBL18945872 0.90 DDB1 (0.75) DDB1CRBNIKZF3TNFIL1B
SCHEMBL283241 0.90 DDB1 (0.75) DDB1CRBNIKZF3TNFIL1B
SCHEMBL18904277 0.90 DDB1 (0.75) DDB1CRBNIKZF3TNFIL1B
Hydrochloric Acid SCHEMBL284302 0.89 DDB1 (0.74) DDB1CRBNIKZF3TNFIL1B
Hydrochloric Acid SCHEMBL284301 0.88 DDB1 (0.72) DDB1CRBNIKZF3TNFIL1B
SCHEMBL18900455 0.86 CRBN (0.80) DDB1CRBNIKZF3TNFIL1B
SCHEMBL18900401 0.81 CRBN (0.49) DDB1CRBNIKZF3TNFIL1B
SCHEMBL25475645 0.81 DDB1 (0.74) DDB1CRBNIKZF3TNFIL1B
SCHEMBL14218469 0.81 DDB1 (0.74) DDB1CRBNIKZF3TNFIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2420498-B1 5-substituted quinazolinone derivatives as anti-cancer agents CELGENE CORP (US) 2017-05-31 EP disclosed
EP-2420498-A1 5-substituted quinazolinone derivatives as anti-cancer agents Celgene Corporation (US) 2012-02-22 EP disclosed