SCHEMBL18945872

SCHEMBL18945872

Cc1nc2cccc(CN)c2c(=O)n1[C@H]1CCC(=O)NC1=O

nearest known ligand 0.75

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
DDB1 Q16531 19/20 0.75
CRBN Q96SW2 19/20 0.75
IKZF3 Q9UKT9 4/20 0.75
TNF P01375 2/20 0.75
IL1B P01584 2/20 0.75
TBXA2R P21731 1/20 0.40
IKZF1 Q13422 1/20 0.40
ALDH1A1 P00352 1/20 0.38
CHRM2 P08172 1/20 0.38
OPRM1 P35372 1/20 0.38
CYP1A2 P05177 1/20 0.38
TSHR P16473 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18904277 1.00 DDB1 (0.75) DDB1CRBNIKZF3TNFIL1B
SCHEMBL283241 1.00 DDB1 (0.75) DDB1CRBNIKZF3TNFIL1B
Hydrochloric Acid SCHEMBL284302 0.99 DDB1 (0.74) DDB1CRBNIKZF3TNFIL1B
Hydrochloric Acid SCHEMBL284301 0.98 DDB1 (0.72) DDB1CRBNIKZF3TNFIL1B
SCHEMBL25475645 0.91 DDB1 (0.74) DDB1CRBNIKZF3TNFIL1B
SCHEMBL14218469 0.91 DDB1 (0.74) DDB1CRBNIKZF3TNFIL1B
SCHEMBL10214943 0.90 DDB1 (0.60) DDB1CRBNIKZF3TNFIL1B
SCHEMBL2603174 0.88 DDB1 (0.70) DDB1CRBNIKZF3TNFIL1B
SCHEMBL24132518 0.88 DDB1 (0.70) DDB1CRBNIKZF3TNFIL1B
SCHEMBL29893790 0.88 DDB1 (0.63) DDB1CRBNIKZF3TNFIL1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11820720-B2 3-(5-substituted-4-oxoquinazolin-3(4H)-yl)-3-deuteropiperidine-2,6-dione derivatives and compositions comprising and methods of using the same SALARIUS PHARMACEUTICALS, INC. (US) 2023-11-21 US disclosed
US-11040925-B2 3-(5-substituted-4-oxoquinazolin-3(4H)-yl)-3-deutero-piperidine-2,6-dione derivatives and compositions comprising and methods of using the same DEUTERX, LLC (US) 2021-06-22 US disclosed
US-20190330124-A1 3-(5-SUBSTITUTED-4-OXOQUINAZOLIN-3(4H)-YL)-3-DEUTERO-PIPERIDINE-2,6-DIONE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SALARIUS PHARMACEUTICALS, INC. 2019-10-31 US disclosed
US-10202316-B2 3-(5-substituted-4-oxoquinazolin-3(4H)-yl)-3-deutero-piperidine-2,6-dione derivatives and compositions comprising and methods of using the same DEUTERX, LLC (US) 2019-02-12 US disclosed
US-20170158579-A1 3-(5-SUBSTITUTED-4-OXOQUINAZOLIN-3(4H)-YL)-3-DEUTERO-PIPERIDINE-2,6-DIONE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME SALARIUS PHARMACEUTICALS, INC. 2017-06-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11820720-B2 3-(5-substituted-4-oxoquinazolin-3(4H)-yl)-3-deuteropiperidine-2,6-dione derivatives and compositions comprising and methods of using the same IL5, IL15, CXCR5 DDB1 781/4885CRBN 2228/4885IKZF3 14/4885
US-11040925-B2 3-(5-substituted-4-oxoquinazolin-3(4H)-yl)-3-deutero-piperidine-2,6-dione derivatives and compositions comprising and methods of using the same IL5, TLR5, IDO1 DDB1 1162/4885CRBN 1871/4885IKZF3 9/4885
US-20190330124-A1 3-(5-SUBSTITUTED-4-OXOQUINAZOLIN-3(4H)-YL)-3-DEUTERO-PIPERIDINE-2,6-DIONE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME IL5, TLR5, IDO1 DDB1 1162/4885CRBN 1871/4885IKZF3 9/4885
US-20170158579-A1 3-(5-SUBSTITUTED-4-OXOQUINAZOLIN-3(4H)-YL)-3-DEUTERO-PIPERIDINE-2,6-DIONE DERIVATIVES AND COMPOSITIONS COMPRISING AND METHODS OF USING THE SAME IL5, TLR5, IDO1 DDB1 1162/4885CRBN 1871/4885IKZF3 9/4885
US-10202316-B2 3-(5-substituted-4-oxoquinazolin-3(4H)-yl)-3-deutero-piperidine-2,6-dione derivatives and compositions comprising and methods of using the same IL5, TLR5, IDO1 DDB1 1162/4885CRBN 1871/4885IKZF3 9/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.