SCHEMBL1022552

SCHEMBL1022552

O=C(NO)OC1c2ccc(OCCN3CCCCC3)cc2CCN1S(=O)(=O)c1ccc(Oc2ccc(F)cc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR1 P03372 5/20 0.51
ESR2 Q92731 5/20 0.51
LTA4H P09960 1/20 0.45
MMP1 P03956 4/20 0.44
MMP7 P09237 4/20 0.44
MMP2 P08253 4/20 0.44
MMP9 P14780 4/20 0.44
MMP12 P39900 3/20 0.44
MMP14 P50281 3/20 0.44
MMP15 P51511 3/20 0.44
MMP16 P51512 3/20 0.44
MMP26 Q9NRE1 3/20 0.44
HTR6 P50406 2/20 0.44
MMP3 P08254 2/20 0.44
HTR1A P08908 1/20 0.44
DRD2 P14416 1/20 0.44
HTR7 P34969 1/20 0.44
HRH3 Q9Y5N1 4/20 0.43
CACNA1B Q00975 2/20 0.42
HDAC3 O15379 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1021934 0.92 EPHX2 (0.46) ESR1ESR2MMP1MMP7MMP2
SCHEMBL1021277 0.92 MMP1 (0.53) ESR1ESR2MMP1MMP7MMP2
SCHEMBL1021841 0.91 ESR1 (0.55) ESR1ESR2LTA4HMMP1MMP7
SCHEMBL1021326 0.91 ESR1 (0.51) ESR1ESR2LTA4HMMP1MMP7
SCHEMBL1020938 0.88 MMP1 (0.43) ESR1ESR2LTA4HMMP1MMP7
SCHEMBL1021428 0.88 MMP1 (0.49) MMP1MMP7MMP2MMP9MMP12
SCHEMBL1022551 0.87 MMP1 (0.58) ESR1ESR2LTA4HMMP1MMP7
SCHEMBL1021990 0.86 CACNA1B (0.43) MMP1MMP7MMP2MMP9MMP12
SCHEMBL1021470 0.85 MMP1 (0.45) MMP1MMP7MMP2MMP9MMP12
SCHEMBL1021839 0.84 ESR1 (0.54) ESR1ESR2LTA4HMMP1MMP7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1869001-B1 SUBSTITUTED TETRAHYDROISOCHINOLINES AS MMP INHIBITORS, RELATED PRODUCTION METHOD AND USE AS MEDICINE SANOFI AVENTIS (FR) 2011-01-12 EP disclosed