SCHEMBL10227481

SCHEMBL10227481

CCc1ccc(-c2ncccc2C#N)cc1

nearest known ligand 0.58

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.58
CYP1A2 P05177 2/20 0.58
CYP2D6 P10635 2/20 0.58
CYP2C9 P11712 2/20 0.58
CYP2C19 P33261 2/20 0.58
CYP3A4 P08684 1/20 0.58
TRPV1 Q8NER1 1/20 0.47
CNR2 P34972 1/20 0.47
HDAC1 Q13547 1/20 0.45
ALDH1A1 P00352 3/20 0.44
L3MBTL1 Q9Y468 3/20 0.44
NPC1 O15118 3/20 0.44
RAB9A P51151 3/20 0.44
SMN1; SMN2 Q16637 3/20 0.44
CASP3 P42574 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
SENP8 Q96LD8 1/20 0.44
SENP7 Q9BQF6 1/20 0.44
SENP6 Q9GZR1 1/20 0.44
SCN9A Q15858 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7683450 0.84 CNR2 (0.47) HPGDCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL8312174 0.83 TRPV1 (0.44) HPGDCYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL7675508 0.81 TRPV1 (0.50) TRPV1CNR2HDAC1SMN1; SMN2SCN9A
SCHEMBL17116613 0.80 CNR2 (0.51) HPGDTRPV1CNR2HDAC1ALDH1A1
SCHEMBL1146096 0.79 HDAC1 (0.51) HPGDTRPV1CNR2HDAC1ALDH1A1
SCHEMBL29768457 0.79 HDAC1 (0.51) HPGDTRPV1CNR2HDAC1ALDH1A1
SCHEMBL24185307 0.78 CNR2 (0.50) HPGDTRPV1CNR2HDAC1ALDH1A1
SCHEMBL18461458 0.78 HDAC1 (0.51) HPGDTRPV1CNR2HDAC1ALDH1A1
SCHEMBL21283226 0.78 CNR2 (0.50) CYP1A2CYP2C9CYP2C19CYP3A4TRPV1
SCHEMBL2471399 0.78 ESR2 (0.53) HPGDTRPV1CNR2HDAC1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8114893-B2 Compounds and methods of use GENENTECH, INC. (US) 2012-02-14 US disclosed