SCHEMBL10229094

SCHEMBL10229094

CCc1[nH]c(=O)c2cc(F)ccc2c1CN1CC=C(c2ccccc2)CC1

nearest known ligand 0.52

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 12/20 0.52
KDM4E B2RXH2 5/20 0.49
MAPT P10636 4/20 0.49
MEN1 O00255 2/20 0.49
KMT2A Q03164 2/20 0.49
CASP1 P29466 1/20 0.48
HBB P68871 1/20 0.48
GAA P10253 4/20 0.47
ALDH1A1 P00352 3/20 0.43
HTT P42858 1/20 0.43
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1720425 0.88 PARP1 (0.54) PARP1KDM4EMAPTMEN1KMT2A
SCHEMBL1721096 0.80 PARP1 (0.43) PARP1KDM4EMAPTMEN1KMT2A
SCHEMBL1719564 0.76 HTR6 (0.56) PARP1KDM4EMAPTMEN1KMT2A
SCHEMBL1721180 0.76 PARP1 (0.61) PARP1KDM4EMAPTMEN1KMT2A
SCHEMBL1720655 0.75 MCL1 (0.41) PARP1ALDH1A1
SCHEMBL10227704 0.74 PARP1 (0.43) PARP1KDM4E
SCHEMBL1720570 0.73 CYP19A1 (0.42) PARP1KDM4EALDH1A1POLB
SCHEMBL1720059 0.73 CYP19A1 (0.42) PARP1KDM4EALDH1A1POLB
SCHEMBL1720056 0.73 CYP19A1 (0.42) PARP1KDM4EALDH1A1POLB
SCHEMBL2564576 0.72 HTR6 (0.53) PARP1MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1566380-B1 ISOQUINOLINE COMPOUNDS AND MEDICINAL USE THEREOF MITSUBISHI TANABE PHARMA CORP (JP) 2012-01-11 EP disclosed