SCHEMBL10232192

SCHEMBL10232192

c1nc(N2CCCCCC3(CC3)C2)c2cc[nH]c2n1

nearest known ligand 0.72

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
JAK3 P52333 17/20 0.72
LCK P06239 3/20 0.57
HTR2C P28335 1/20 0.56
DOT1L Q8TEK3 1/20 0.55
AKT2 P31751 1/20 0.54
GSK3B P49841 1/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20470386 0.95 JAK3 (0.69) JAK3LCKHTR2CDOT1LAKT2
SCHEMBL2018963 0.85 JAK3 (1.00) JAK3LCKHTR2CDOT1LAKT2
SCHEMBL3959075 0.85 JAK3 (1.00) JAK3LCKHTR2CDOT1LAKT2
SCHEMBL1048998 0.85 JAK3 (1.00) JAK3LCKHTR2CDOT1LAKT2
SCHEMBL1818852 0.83 JAK3 (1.00) JAK3LCKHTR2CDOT1LAKT2
SCHEMBL323332 0.81 HTR2C (0.69) JAK3LCKHTR2CDOT1LAKT2
SCHEMBL10206799 0.81 JAK3 (0.83) JAK3LCKHTR2CDOT1L
SCHEMBL2021631 0.81 JAK3 (0.68) JAK3LCK
SCHEMBL31550436 0.80 JAK3 (0.93) JAK3LCKHTR2CDOT1LAKT2
SCHEMBL29073290 0.80 AKT2 (0.68) JAK3LCKHTR2CDOT1LAKT2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012003829-A1 NOVEL HOMOPIPERAZINE DERIVATIVES AS PROTEIN TYROSINE KINASE INHIBITORS AND PHARMACEUTICAL USE THEREOF LEO PHARMA A/S (DK) 2012-01-12 WO disclosed