SCHEMBL10240546

SCHEMBL10240546

Bc1ccc(C)cc1S(=O)(=O)Nc1ccc2c(c1)CCN(C(=O)OC(C)(C)C)C2

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.54
KCNA1 Q09470 4/20 0.48
KCNAB1 Q14722 4/20 0.48
NR1H2 P55055 1/20 0.48
LMNA P02545 2/20 0.44
CYP1A2 P05177 1/20 0.44
CYP3A4 P08684 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
RECQL P46063 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
NAMPT P43490 2/20 0.43
PTPN1 P18031 2/20 0.41
TMPRSS2 O15393 1/20 0.41
IGF1R P08069 1/20 0.41
KIT P10721 1/20 0.40
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3156959 0.88 SMN1; SMN2 (0.54) ESR2KCNA1KCNAB1LMNAJAK2
SCHEMBL4789781 0.83 ESR2 (0.66) ESR2KCNA1KCNAB1NR1H2NPC1
SCHEMBL2056208 0.81 ESR2 (0.76) ESR2NR1H2NPC1RAB9ANAMPT
SCHEMBL3142771 0.80 ESR2 (0.53) ESR2KCNA1KCNAB1NR1H2LMNA
SCHEMBL5600152 0.79 NR1H2 (0.65) ESR2KCNA1KCNAB1NR1H2NPC1
SCHEMBL16645111 0.79 ESR2 (0.60) ESR2KCNA1KCNAB1NR1H2NPC1
SCHEMBL3155935 0.79 ESR2 (0.54) ESR2NR1H2NPC1RAB9ANAMPT
SCHEMBL1187860 0.79 ESR2 (0.62) ESR2KCNA1KCNAB1NR1H2NPC1
SCHEMBL6393284 0.78 PTPN1 (0.64) ESR2KCNA1KCNAB1NR1H2NPC1
SCHEMBL16645108 0.78 ESR2 (0.53) ESR2KCNA1KCNAB1NR1H2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2007729-B1 SUBSTITUTED TETRAHYDROISOQUINOLINE COMPOUNDS, THEIR PREPARATION AND USE IN MEDICAMENTS ESTEVE LABOR DR (ES) 2012-06-27 EP disclosed