SCHEMBL1024327

SCHEMBL1024327

CC(C)(C)N(C(=O)O)c1cccc(NC(=O)c2cccc(N)c2)c1

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PTGS1 P23219 3/20 0.53
KCNK9 Q9NPC2 4/20 0.48
KCNK3 O14649 5/20 0.47
ALDH1A1 P00352 4/20 0.47
KDM4E B2RXH2 1/20 0.47
ULK1 O75385 1/20 0.46
KMT2A Q03164 4/20 0.46
MEN1 O00255 3/20 0.46
POLB P06746 2/20 0.46
KCNH2 Q12809 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
MAPK1 P28482 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.46
SMN1; SMN2 Q16637 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
HSD17B10 Q99714 1/20 0.45
KDM4C Q9H3R0 1/20 0.44
BTK Q06187 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1026693 0.82 ALDH1A1 (0.42) PTGS1ALDH1A1KDM4EKMT2AMEN1
SCHEMBL1026082 0.81 MEN1 (0.63) ALDH1A1KMT2AMEN1POLBRAB9A
SCHEMBL1025671 0.81 NR1H4 (0.48) ALDH1A1KDM4EPOLBHTTRAB9A
SCHEMBL1026084 0.81 MEN1 (0.63) ALDH1A1KMT2AMEN1POLBRAB9A
SCHEMBL1028225 0.80 ALDH1A1 (0.48) ALDH1A1KDM4EKMT2AMEN1POLB
SCHEMBL2126328 0.79 PTGS1 (0.68) PTGS1KCNK9KCNK3ALDH1A1KDM4E
SCHEMBL31171978 0.79 PTGS1 (0.72) PTGS1KCNK9KCNK3ALDH1A1KDM4E
SCHEMBL308208 0.79 PTGS1 (0.72) PTGS1KCNK9KCNK3ALDH1A1KDM4E
SCHEMBL1025733 0.78 ALDH1A1 (0.59) ALDH1A1POLBHTTRAB9A
SCHEMBL1352405 0.78 PTGS1 (0.68) PTGS1KCNK9KCNK3ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274288-A2 MACROCYCLIC COMPOUNDS AND THEIR USE AS KINASE INHIBITORS Incyte Corporation (US) 2011-01-19 EP disclosed