SCHEMBL10248380

SCHEMBL10248380

Nc1ccc(S(=O)(=O)NCc2cccc(CN(Cc3ccc(-c4ccccc4)cc3)S(=O)(=O)c3cc(Cl)cc(Cl)c3O)c2)cc1

nearest known ligand 0.66

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ACLY P53396 9/20 0.66
CYP19A1 P11511 1/20 0.44
MMP1 P03956 1/20 0.43
MMP2 P08253 1/20 0.43
MMP9 P14780 1/20 0.43
MMP8 P22894 1/20 0.43
MMP13 P45452 1/20 0.43
CA12 O43570 2/20 0.43
CA1 P00915 2/20 0.43
CA2 P00918 2/20 0.43
CA4 P22748 2/20 0.43
CA9 Q16790 2/20 0.43
BCL2 P10415 1/20 0.43
CXCR3 P49682 1/20 0.41
PDK1 Q15118 1/20 0.41
TAS2R14 Q9NYV8 1/20 0.40
LMNA P02545 1/20 0.40
SLC12A2 P55011 1/20 0.40
SLC12A5 Q9H2X9 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL252751 0.94 ACLY (0.71) ACLYCYP19A1MMP1MMP2MMP9
SCHEMBL183817 0.92 ACLY (0.66) ACLYCYP19A1MMP1MMP2MMP9
SCHEMBL184772 0.91 ACLY (0.70) ACLYCYP19A1MMP1MMP2MMP9
SCHEMBL184516 0.91 ACLY (0.65) ACLYMMP1MMP2MMP9MMP8
SCHEMBL184807 0.90 ACLY (0.74) ACLYMMP1MMP2MMP9MMP8
SCHEMBL15157462 0.90 ACLY (0.64) ACLYCYP19A1MMP1MMP2MMP9
SCHEMBL10248987 0.90 ACLY (0.68) ACLYMMP1MMP2MMP9MMP8
SCHEMBL253454 0.89 ACLY (0.62) ACLYCYP19A1MMP1MMP2MMP9
SCHEMBL184201 0.89 ACLY (0.65) ACLYCYP19A1MMP1MMP2MMP9
SCHEMBL184198 0.87 ACLY (0.61) ACLYMMP1MMP2MMP9MMP8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297103-B1 HYDROXYPHENYLSULFONAMIDES AS ANTIAPOPTOTIC BCL INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2012-01-04 EP disclosed