SCHEMBL10248875

SCHEMBL10248875

O=C(NCc1cccc(CN(Cc2ccc(C(F)(F)F)cc2)S(=O)(=O)c2cc(Cl)cc(Cl)c2O)c1)NC1CC=C(F)C=C1F

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACLY P53396 2/20 0.46
BCL2 P10415 1/20 0.42
MMP1 P03956 1/20 0.38
MMP2 P08253 1/20 0.38
MMP9 P14780 1/20 0.38
MMP8 P22894 1/20 0.38
MMP13 P45452 1/20 0.38
TRPV1 Q8NER1 7/20 0.37
CXCR3 P49682 2/20 0.36
KCNH2 Q12809 1/20 0.34
MCHR1 Q99705 1/20 0.34
MAPT P10636 1/20 0.34
MEN1 O00255 1/20 0.34
PLA2G1B P04054 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
GAA P10253 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL184590 0.82 ACLY (0.59) ACLYBCL2MMP1MMP2MMP9
SCHEMBL183990 0.79 BCL2 (0.48) ACLYBCL2MMP1MMP2MMP9
SCHEMBL184862 0.79 ACLY (0.52) ACLYBCL2MMP1MMP2MMP9
SCHEMBL185069 0.79 ACLY (0.60) ACLYBCL2MMP1MMP2MMP9
SCHEMBL184826 0.76 ACLY (0.61) ACLYBCL2MMP1MMP2MMP9
SCHEMBL2734939 0.75 ACLY (0.49) ACLYBCL2MMP1MMP2MMP9
SCHEMBL254105 0.75 ACLY (0.62) ACLYBCL2MMP1MMP2MMP9
SCHEMBL184743 0.74 BCL2 (0.64) ACLYBCL2MMP1MMP2MMP9
SCHEMBL184004 0.74 ACLY (0.47) ACLYBCL2MMP1MMP2MMP9
SCHEMBL184298 0.73 ACLY (0.74) ACLYBCL2MMP1MMP2MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2297103-B1 HYDROXYPHENYLSULFONAMIDES AS ANTIAPOPTOTIC BCL INHIBITORS BRISTOL MYERS SQUIBB CO (US) 2012-01-04 EP disclosed