SCHEMBL10249426

SCHEMBL10249426

O=C[C@H](CC(=O)O)NC(=O)CN1C(=O)C(NC(=O)c2cccc3ccccc23)CN(C=O)c2ccccc21

nearest known ligand 0.52

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 11/20 0.52
IL1B P01584 1/20 0.39
XIAP P98170 7/20 0.39
CCKBR P32239 1/20 0.38
CYP3A4 P08684 2/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12444043 1.00 CASP1 (0.52) CASP1IL1BXIAPCCKBRCYP3A4
SCHEMBL647286 1.00 CASP1 (0.52) CASP1IL1BXIAPCCKBRCYP3A4
SCHEMBL12443659 0.93 CASP1 (0.45) CASP1XIAPCYP3A4
SCHEMBL10251968 0.93 CASP1 (0.45) CASP1XIAPCYP3A4
SCHEMBL10200303 0.93 CASP1 (0.45) CASP1XIAPCYP3A4
SCHEMBL10199304 0.89 CASP1 (0.53) CASP1XIAPCYP3A4
SCHEMBL10201335 0.87 CASP1 (0.52) CASP1XIAPCYP3A4
SCHEMBL10263997 0.86 CASP1 (0.52) CASP1XIAPCYP3A4
SCHEMBL644733 0.85 CASP1 (0.50) CASP1XIAPCYP3A4
SCHEMBL10284695 0.85 CASP1 (0.49) CASP1XIAPCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119631-B2 Inhibitors of interleukin-1β converting enzyme VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-21 US disclosed
US-8119631-B2 Inhibitors of interleukin-1β converting enzyme VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-21 US disclosed