SCHEMBL10255307

SCHEMBL10255307

COC(=O)N1CCN(c2cncc(-c3nnc(-c4ccccc4)o3)n2)CC1

nearest known ligand 0.49

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 6/20 0.49
ATR Q13535 2/20 0.45
CKS1B P61024 4/20 0.44
SKP1 P63208 4/20 0.44
SKP2 Q13309 4/20 0.44
PIM2 Q9P1W9 6/20 0.44
PIM1 P11309 1/20 0.41
CSNK2A2 P19784 1/20 0.41
CSNK2A1 P68400 1/20 0.41
NPC1 O15118 1/20 0.41
TSHR P16473 1/20 0.41
RAB9A P51151 1/20 0.41
ALOX15 P16050 1/20 0.40
HSD17B10 Q99714 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10255806 0.91 ATR (0.55) DGAT1ATRHSD17B10
SCHEMBL10255790 0.88 ATR (0.47) DGAT1ATRCKS1BSKP1SKP2
SCHEMBL10255318 0.88 PIM2 (0.56) ATRCKS1BSKP1SKP2PIM2
SCHEMBL10255214 0.87 GAA (0.48) ATRCKS1BSKP1SKP2PIM2
SCHEMBL10255313 0.86 ATR (0.47) DGAT1ATRPIM2NPC1RAB9A
SCHEMBL10255788 0.85 NPC1 (0.52) ATRCKS1BSKP1SKP2PIM2
SCHEMBL10255249 0.85 CKS1B (0.57) ATRCKS1BSKP1SKP2PIM2
SCHEMBL10255255 0.85 PIM2 (0.44) ATRCKS1BSKP1SKP2PIM2
SCHEMBL14822722 0.85 NPC1 (0.56) ATRCKS1BSKP1SKP2PIM2
SCHEMBL10256348 0.85 RAB9A (0.50) ATRCKS1BSKP1SKP2PIM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8410112-B2 Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-02 US disclosed
US-20120040020-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120040020-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK2, CHEK1 DGAT1 4471/4885ATR 1/4885CKS1B 117/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.