SCHEMBL10257367

SCHEMBL10257367

CNCc1ccc(-c2nnc(-c3cncc(C4CC4C(=O)NCC(O)CO)n3)o2)cc1

nearest known ligand 0.36

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ATR Q13535 10/20 0.36
S1PR1 P21453 2/20 0.36
SPHK1 Q9NYA1 1/20 0.32
PRMT5 O14744 2/20 0.32
ALDH1A1 P00352 1/20 0.32
CTSK P43235 1/20 0.31
PIM1 P11309 1/20 0.30
PIM3 Q86V86 1/20 0.30
PIM2 Q9P1W9 1/20 0.30
NAMPT P43490 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10256088 0.88 SPHK1 (0.38) ATRSPHK1ALDH1A1CTSKPIM1
SCHEMBL615908 0.85 ATR (0.51) ATR
SCHEMBL10256086 0.77 ATR (0.38) ATRPIM1PIM2
SCHEMBL10256640 0.76 ATR (0.40) ATRSPHK1PIM1PIM3PIM2
SCHEMBL617527 0.73 ATR (0.55) ATR
SCHEMBL10256031 0.70 NAMPT (0.41) ATRALDH1A1PIM1PIM3PIM2
SCHEMBL16420624 0.69 ATR (0.54) ATR
SCHEMBL16420659 0.67 ATR (0.48) ATR
SCHEMBL16489024 0.67 ATR (0.52) ATR
SCHEMBL10256712 0.67 AADAT (0.40) ATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8410112-B2 Compounds useful as inhibitors of ATR kinase VERTEX PHARMACEUTICALS INCORPORATED (US) 2013-04-02 US disclosed
US-20120040020-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE VERTEX PHARMACEUTICALS INCORPORATED (US) 2012-02-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120040020-A1 COMPOUNDS USEFUL AS INHIBITORS OF ATR KINASE ATR, CHEK2, CHEK1 ATR 1/4885S1PR1 2774/4885SPHK1 1417/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.