SCHEMBL1025923

SCHEMBL1025923

N[C@@H](CO)C(=O)NCCN(Cc1ccccc1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
REN P00797 2/20 0.47
CNR1 P21554 1/20 0.43
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
MMP2 P08253 1/20 0.41
CYP3A4 P08684 1/20 0.40
TSHR P16473 1/20 0.40
HDAC8 Q9BY41 1/20 0.40
MC4R P32245 1/20 0.39
MC5R P33032 1/20 0.39
MC3R P41968 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5183620 1.00 REN (0.47) RENCNR1CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL4847760 0.99 REN (0.46) RENCNR1CYP2D6CYP2C9CYP2C19
SCHEMBL1021811 0.80 SLC1A3 (0.56)
SCHEMBL8054823 0.79 POLB (0.55) CNR1CYP2D6CYP2C9CYP2C19KMT2A
SCHEMBL19710389 0.79 POLB (0.55) CNR1CYP2D6CYP2C9CYP2C19KMT2A
SCHEMBL11884007 0.79 REN (0.57) RENKMT2AALDH1A1NPSR1TSHR
Hydrochloric Acid SCHEMBL4854908 0.79 SLC1A3 (0.55)
Hydrochloric Acid SCHEMBL11100779 0.78 CYP2D6 (0.63) CNR1CYP2D6CYP2C9CYP2C19KMT2A
Hydrochloric Acid SCHEMBL20569304 0.77 KMT2A (0.57) CNR1CYP2D6CYP2C9CYP2C19KMT2A
Hydrochloric Acid SCHEMBL20569306 0.77 KMT2A (0.57) CNR1CYP2D6CYP2C9CYP2C19KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1797110-B1 ANTIBACTERIAL AMIDE MACROCYCLES IV AICURIS GMBH & CO KG (DE) 2011-01-12 EP disclosed
EP-1797110-A1 ANTIBACTERIAL AMIDE MACROCYCLES IV AiCuris GmbH & Co. KG (DE) 2007-06-20 EP disclosed
WO-2006034786-A1 ANTIBACTERIAL AMIDE MACROCYCLES IV AICURIS GMBH & CO.KG (DE) 2006-04-06 WO disclosed