SCHEMBL10270159

SCHEMBL10270159

Cc1nc(-c2ccc(Cl)cc2Cl)cc2nc(CN3CCCCC3)nn12

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 1/20 0.42
CRHR1 P34998 3/20 0.41
DPP4 P27487 10/20 0.41
DPP8 Q6V1X1 6/20 0.41
DPP9 Q86TI2 5/20 0.41
OPRL1 P41146 1/20 0.41
CYP3A4 P08684 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
CNR1 P21554 2/20 0.38
CNR2 P34972 2/20 0.38
HSP90AA1 P07900 1/20 0.38
HSP90AB1 P08238 1/20 0.38
ACP1 P24666 1/20 0.38
PDE10A Q9Y233 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12680488 0.89 CNR1 (0.39) SIGMAR1CRHR1DPP4DPP8DPP9
SCHEMBL12680458 0.87 ALPL (0.41) SIGMAR1CRHR1DPP4DPP8DPP9
SCHEMBL3611015 0.78 CYP2A13 (0.47) SIGMAR1CRHR1DPP4DPP8DPP9
SCHEMBL3607437 0.77 CYP2A13 (0.45) SIGMAR1CRHR1DPP4
SCHEMBL10270029 0.76 GSK3B (0.36) SIGMAR1DPP4DPP8DPP9CYP3A4
SCHEMBL10269950 0.76 HRH4 (0.37) SIGMAR1DPP4DPP8DPP9CNR1
SCHEMBL10270288 0.75 DPP4 (0.39) CRHR1DPP4DPP8DPP9CYP3A4
SCHEMBL12680882 0.74 GSK3B (0.48) DPP4DPP8CNR1CNR2
SCHEMBL12680879 0.73 CNR1 (0.35) SIGMAR1DPP4DPP8DPP9CNR1
SCHEMBL12680493 0.69 CYP1A2 (0.41) SIGMAR1CRHR1DPP4DPP8DPP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2137188-B1 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES Bayer Pharma AG (DE) 2012-06-06 EP disclosed
WO-2008113469-A2 SUBSTITUTED IMIDAZOPYRIMIDINES AND TRIAZOLOPYRIMIDINES BAYER SCHERING PHARMA AKTIENGESELLSCHAFT (DE) 2008-09-25 WO disclosed