SCHEMBL10272089

SCHEMBL10272089

CC[C@@H](Nc1nc(Nc2cccc(OC(F)F)c2)c(C(N)=O)c(=O)[nH]1)C(N)=O

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
SYK P43405 13/20 0.43
EP300 Q09472 1/20 0.39
CREBBP Q92793 1/20 0.39
MLKL Q8NB16 1/20 0.39
PIK3CA P42336 1/20 0.39
GRM4 Q14833 2/20 0.39
TAS2R14 Q9NYV8 1/20 0.38
BUB1 O43683 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2718425 0.91 SYK (0.44) SYK
SCHEMBL2718419 0.91 SYK (0.44) SYK
SCHEMBL10271735 0.91 SYK (0.42) SYK
SCHEMBL2715960 0.91 SYK (0.52) SYKMLKLPIK3CA
SCHEMBL10272215 0.87 SYK (0.45) SYK
SCHEMBL2716538 0.86 SYK (0.50) SYK
SCHEMBL2715926 0.82 SYK (0.42) SYK
SCHEMBL2715928 0.82 SYK (0.42) SYK
SCHEMBL2716671 0.82 SYK (0.51) SYKMLKL
SCHEMBL2716675 0.82 SYK (0.51) SYKMLKL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012061415-A1 OXYPYRIMIDINES AS SYK MODULATORS PORTOLA PHARMACEUTICALS, INC. (US) 2012-05-10 WO disclosed