SCHEMBL10272808

SCHEMBL10272808

CCc1ccc(C(C)(C)OCOC)nc1

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADORA2A P29274 1/20 0.38
HDAC1 Q13547 1/20 0.38
KDM4E B2RXH2 2/20 0.35
L3MBTL1 Q9Y468 2/20 0.35
PDE10A Q9Y233 1/20 0.32
PTGS2 P35354 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
CYP1A2 P05177 1/20 0.31
CYP2D6 P10635 1/20 0.31
CA2 P00918 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18808193 0.80 CCR1 (0.36) ADORA2AHDAC1KDM4EPDE10A
SCHEMBL2733260 0.79 HDAC1 (0.36) ADORA2AHDAC1KDM4EL3MBTL1NPC1
SCHEMBL16523823 0.79 HDAC1 (0.36) ADORA2AHDAC1
SCHEMBL210170 0.75 HDAC1 (0.35) ADORA2AHDAC1CA2
SCHEMBL1755679 0.75 KDM4E (0.43) KDM4EL3MBTL1PDE10APTGS2NPC1
SCHEMBL30802846 0.75 KDM4E (0.43) KDM4EL3MBTL1PDE10APTGS2NPC1
SCHEMBL10272809 0.72 PDE10A (0.46) KDM4EL3MBTL1PDE10APTGS2NPC1
SCHEMBL15986681 0.72 L3MBTL1 (0.41) KDM4EL3MBTL1PDE10APTGS2NPC1
SCHEMBL16368521 0.72 KDM4E (0.41) KDM4EL3MBTL1PDE10APTGS2NPC1
SCHEMBL12266677 0.72 KDM4E (0.41) KDM4EL3MBTL1PDE10APTGS2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8088805-B2 Inhibitors of histone deacetylase METHYLGENE INC. (CA) 2012-01-03 US disclosed