SCHEMBL10274785

SCHEMBL10274785

CN(C)C1CCN(c2ccc3cnccc3c2)CC1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PHGDH O43175 1/20 0.45
CYP19A1 P11511 1/20 0.44
CDK4 P11802 15/20 0.43
CDK6 Q00534 7/20 0.43
CDK1 P06493 3/20 0.43
CCNB1 P14635 3/20 0.43
CCND1 P24385 3/20 0.43
CCND3 P30281 2/20 0.43
FLT3 P36888 2/20 0.41
HRH3 Q9Y5N1 1/20 0.40
MKNK2 Q9HBH9 1/20 0.40
CCNA2 P20248 1/20 0.40
CDK2 P24941 1/20 0.40
CCNA1 P78396 1/20 0.40
KIT P10721 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL803946 0.82 KDM4E (0.51) PHGDHHRH3
SCHEMBL803705 0.81 F10 (0.43) PHGDH
SCHEMBL803945 0.79 PDE10A (0.44) PHGDH
SCHEMBL30738297 0.79 CYP19A1 (0.54) PHGDHCYP19A1MKNK2
SCHEMBL15516206 0.79 CYP19A1 (0.54) PHGDHCYP19A1MKNK2
SCHEMBL2362576 0.77 CHKA (0.53) FLT3HRH3KIT
SCHEMBL6017418 0.75 HTR3E (0.63) PHGDHCYP19A1
SCHEMBL22837854 0.75 NPY5R (0.53) HRH3
Hydrochloric Acid SCHEMBL30609660 0.74 HTR3E (0.61) PHGDHCYP19A1
Hydrochloric Acid SCHEMBL2801289 0.74 HTR3E (0.61) PHGDHCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012038081-A1 SUBSTITUTED BENZAMIDE COMPOUNDS Grünenthal GmbH (DE) 2012-03-29 WO disclosed