SCHEMBL10279853

SCHEMBL10279853

COCC(=O)NC(C)COc1ccc2c(cnn2-c2ccc(F)cc2)c1

nearest known ligand 0.60

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 19/20 0.60
PGR P06401 3/20 0.52
SMO Q99835 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10280471 0.82 NR3C1 (0.59) NR3C1PGRSMO
SCHEMBL837296 0.81 NR3C1 (0.84) NR3C1PGR
SCHEMBL837295 0.81 NR3C1 (0.84) NR3C1PGR
SCHEMBL833507 0.80 NR3C1 (0.74) NR3C1PGR
SCHEMBL833506 0.80 NR3C1 (0.74) NR3C1PGR
SCHEMBL836800 0.80 NR3C1 (0.69) NR3C1PGR
SCHEMBL836799 0.80 NR3C1 (0.69) NR3C1PGR
SCHEMBL835417 0.80 NR3C1 (0.66) NR3C1PGR
SCHEMBL835418 0.80 NR3C1 (0.66) NR3C1PGR
SCHEMBL836283 0.79 NR3C1 (0.68) NR3C1PGR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2102169-B1 INDAZOLYL AMIDE DERIVATIVES FOR THE TREATMENT OF GLUCOCORTICOID RECEPTOR MEDIATED DISORDERS ASTRAZENECA AB (SE) 2012-06-20 EP disclosed