SCHEMBL10280429

SCHEMBL10280429

COBNCC1CCN(c2cc(C(=O)Nc3ccccc3)ccc2[N+](=O)[O-])CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TAAR1 Q96RJ0 1/20 0.51
ALDH1A1 P00352 11/20 0.49
TDP1 Q9NUW8 2/20 0.49
CYP3A4 P08684 1/20 0.49
TSHR P16473 1/20 0.49
MAPT P10636 7/20 0.47
SMN1; SMN2 Q16637 4/20 0.47
MAPK1 P28482 2/20 0.47
LMNA P02545 2/20 0.47
KMT2A Q03164 6/20 0.46
MEN1 O00255 5/20 0.46
GAA P10253 1/20 0.46
NPC1 O15118 2/20 0.45
RAB9A P51151 2/20 0.45
HTT P42858 1/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
NPSR1 Q6W5P4 1/20 0.44
CASP3 P42574 1/20 0.43
SENP7 Q9BQF6 1/20 0.43
POLB P06746 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10280428 0.86 IRAK1 (0.45) TAAR1ALDH1A1TDP1MAPTNPC1
SCHEMBL10259263 0.84 TAAR1 (0.49) TAAR1ALDH1A1TDP1CYP3A4TSHR
SCHEMBL358097 0.83 TAAR1 (0.49) TAAR1ALDH1A1TDP1CYP3A4TSHR
SCHEMBL28954877 0.71 TAAR1 (0.58) TAAR1ALDH1A1TDP1CYP3A4TSHR
SCHEMBL358680 0.69 ALDH1A1 (0.81) ALDH1A1TDP1CYP3A4TSHRMAPT
SCHEMBL10254666 0.69 IRAK1 (0.46) ALDH1A1TDP1MAPT
SCHEMBL358342 0.69 ACACB (0.51)
SCHEMBL8303947 0.69 ALDH1A1 (0.71) ALDH1A1TDP1CYP3A4TSHRMAPT
SCHEMBL16146269 0.69 IRAK1 (0.60) ALDH1A1MAPTSMN1; SMN2NPC1RAB9A
SCHEMBL3645707 0.68 TAAR1 (1.00) TAAR1ALDH1A1MAPTSMN1; SMN2MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012007375-A1 PYRAZOLO [1, 5A] PYRIMIDINE AND THIENO [3, 2B] PYRIMIDINE DERIVATIVES AS IRAK4 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2012-01-19 WO disclosed