SCHEMBL10284366

SCHEMBL10284366

C=C(c1ccc(C(=O)NC2CCN(Cc3ccc(C#N)cc3)CC2)cn1)N1CCC(C(=O)c2ccc(OC)cc2)CC1

nearest known ligand 0.86

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PRKAB2 O43741 14/20 0.86
PRKAG1 P54619 14/20 0.86
PRKAA2 P54646 14/20 0.86
PRKAA1 Q13131 14/20 0.86
PRKAG3 Q9UGI9 14/20 0.86
PRKAG2 Q9UGJ0 14/20 0.86
PRKAB1 Q9Y478 14/20 0.86
KCNH2 Q12809 1/20 0.86
CYP3A4 P08684 2/20 0.69

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL517986 0.92 PRKAB2 (1.00) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL518529 0.90 PRKAA2 (0.90) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL518679 0.87 PRKAB2 (0.87) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL518517 0.87 PRKAA2 (1.00) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL16615397 0.86 PRKAA2 (0.89) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL22268945 0.85 PRKAA2 (0.81) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL518740 0.85 PRKAA2 (0.77) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL15171532 0.85 PRKAB2 (0.84) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL518414 0.85 PRKAB2 (0.83) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3
SCHEMBL518887 0.84 PRKAA2 (0.92) PRKAB2PRKAG1PRKAA2PRKAA1PRKAG3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012016217-A1 AMPK-ACTIVATING HETEROCYCLIC COMPOUNDS AND METHODS FOR USING THE SAME RIGEL PHARMACEUTICALS, INC. (US) 2012-02-02 WO disclosed