SCHEMBL1029161

SCHEMBL1029161

COCCCOC(=O)N1CCc2cc(C(=O)NO)ccc2C1

nearest known ligand 0.59

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
HDAC6 Q9UBN7 17/20 0.59
HDAC8 Q9BY41 5/20 0.59
HDAC1 Q13547 2/20 0.53
HDAC3 O15379 1/20 0.53
TMPRSS2 O15393 1/20 0.44
POLB P06746 1/20 0.43
TMEM97 Q5BJF2 1/20 0.43
SIGMAR1 Q99720 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1073298 0.95 HDAC6 (0.54) HDAC6HDAC8HDAC1HDAC3
SCHEMBL2277596 0.83 HDAC6 (0.58) HDAC6HDAC8HDAC1HDAC3POLB
SCHEMBL1027140 0.80 HDAC6 (0.62) HDAC6HDAC8HDAC1HDAC3
SCHEMBL1082437 0.80 TMEM97 (0.64) HDAC6HDAC8HDAC1HDAC3TMEM97
SCHEMBL2275604 0.79 HDAC6 (0.42) HDAC6HDAC8TMPRSS2POLBTMEM97
SCHEMBL2283261 0.79 HDAC6 (0.53) HDAC6HDAC8HDAC1HDAC3POLB
SCHEMBL1027560 0.78 HDAC6 (0.73) HDAC6HDAC8HDAC1HDAC3
SCHEMBL1081445 0.75 HDAC6 (0.70) HDAC6HDAC8HDAC1HDAC3TMPRSS2
SCHEMBL8264660 0.75 ABHD6 (0.56) POLBTMEM97SIGMAR1
SCHEMBL2283593 0.75 MAP3K5 (0.39) HDAC6TMEM97SIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2274283-A1 NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS 4SC AG (DE) 2011-01-19 EP disclosed
WO-2009112550-A1 NOVEL N-SUBSTITUTED TETRAHYDROISOQUINOLINE/ISOINDOLINE HYDROXAMIC ACID COMPOUNDS 4SC AG (DE) 2009-09-17 WO disclosed