SCHEMBL10293824

SCHEMBL10293824

NS(=O)(=O)OC[C@H]1CCC(n2ccc3c(NCc4ccccc4Cl)ncnc32)C1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAE1 Q13564 6/20 0.48
UBA3 Q8TBC4 5/20 0.48
CA2 P00918 2/20 0.48
SAE1 Q9UBE0 2/20 0.48
UBA2 Q9UBT2 2/20 0.48
GRK5 P34947 1/20 0.48
CSNK1A1 P48729 1/20 0.48
UBA6 A0AVT1 1/20 0.48
NEDD8 Q15843 1/20 0.48
AURKA O14965 1/20 0.42
RPS6KB1 P23443 1/20 0.42
LMNA P02545 3/20 0.40
ALDH1A1 P00352 2/20 0.40
PKM P14618 1/20 0.40
PIP4K2A P48426 1/20 0.40
KDM4E B2RXH2 1/20 0.39
MAPK1 P28482 1/20 0.39
ADORA3 P0DMS8 1/20 0.38
ADORA2A P29274 1/20 0.38
ADORA1 P30542 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2740570 0.90 NAE1 (0.44) NAE1UBA3CA2SAE1UBA2
SCHEMBL2740588 0.89 NAE1 (0.48) NAE1UBA3CA2SAE1UBA2
SCHEMBL10235267 0.88 NAE1 (0.47) NAE1UBA3CA2SAE1UBA2
SCHEMBL10293821 0.88 NAE1 (0.51) NAE1UBA3CA2SAE1UBA2
SCHEMBL10293816 0.88 NAE1 (0.47) NAE1UBA3CA2SAE1UBA2
SCHEMBL10233932 0.86 CA2 (0.46) NAE1UBA3CA2SAE1UBA2
SCHEMBL13192031 0.86 NAE1 (0.44) NAE1UBA3CA2SAE1UBA2
SCHEMBL10242205 0.86 NAE1 (0.49) NAE1UBA3CA2SAE1UBA2
SCHEMBL10236878 0.85 NAE1 (0.43) NAE1UBA3CA2SAE1UBA2
SCHEMBL191795 0.85 NAE1 (0.65) NAE1UBA3CA2SAE1UBA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1989206-B1 INHIBITORS OF E1 ACTIVATING ENZYME MILLENNIUM PHARM INC (US) 2012-07-04 EP disclosed