SCHEMBL10299593

SCHEMBL10299593

COC(=O)C(N)N

nearest known ligand 0.00

⚠ Novel chemotype — no close known analogue (best Tanimoto < 0.3). Unexplored chemical space relative to ChEMBL.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Acetic Acid SCHEMBL28778977 0.91 SMN1; SMN2 (0.42)
SCHEMBL279148 0.80 SMN1; SMN2 (0.48)
Hydrochloric Acid SCHEMBL655143 0.78 SMN1; SMN2 (0.46)
SCHEMBL16081670 0.78
SCHEMBL10151193 0.78
SCHEMBL41892 0.78
SCHEMBL30039818 0.78
SCHEMBL104803 0.78
SCHEMBL72838 0.78
SCHEMBL25301326 0.75

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4209498-A1 4'-THIO-NUCLEOTIDE AND -NUCLEOSIDE PRODRUGS FOR THE TREATMENT OF CANCER Southern Research Institute (US) 2023-07-12 EP disclosed
US-20230133817-A1 MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS RQX PHARMACEUTICALS INC (US) 2023-05-04 US disclosed
US-20210198316-A9 MACROCYCLIC BROAD SPECTRUM ANTIBIOTICS CHARLES RIVER DISCOVERY RESEARCH SERVICES UK LIMITED (GB) 2021-07-01 US disclosed
WO-2017114382-A1 METHOD FOR SYNTHESIZING C-TERMINAL MODIFIED PEPTIDE 深圳翰宇药业股份有限公司 2017-07-06 WO disclosed
US-8217031-B2 Heteroaryl derivatives NIPPON SHINYAKU CO., LTD. (JP) 2012-07-10 US disclosed
US-20100048537-A1 HETEROARYL DERIVATIVES NIPPON SHINYAKU CO., LTD. (JP) 2010-02-25 US disclosed