SCHEMBL103123

SCHEMBL103123

CNC(=O)c1ccc(Cl)nc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 6/20 0.61
SMN1; SMN2 Q16637 3/20 0.61
NAPRT Q6XQN6 1/20 0.60
KMT2A Q03164 4/20 0.56
NPC1 O15118 3/20 0.56
MEN1 O00255 3/20 0.56
POLB P06746 1/20 0.56
BAZ2B Q9UIF8 1/20 0.56
L3MBTL1 Q9Y468 1/20 0.55
EGFR P00533 2/20 0.54
TDP1 Q9NUW8 1/20 0.54
MDM4 O15151 1/20 0.54
TP53 P04637 1/20 0.54
MDM2 Q00987 1/20 0.54
ALDH1A1 P00352 2/20 0.54
LMNA P02545 1/20 0.54
GAA P10253 2/20 0.53
MAPT P10636 1/20 0.52
PKM P14618 1/20 0.52
KCNQ3 O43525 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL29989142 0.87 RAB9A (0.56) RAB9ASMN1; SMN2NAPRTKMT2ANPC1
SCHEMBL13184552 0.82 BAZ2B (0.57) RAB9ASMN1; SMN2KMT2ANPC1MEN1
SCHEMBL1725139 0.82 NAPRT (0.62) RAB9ASMN1; SMN2NAPRTKMT2ANPC1
SCHEMBL31295356 0.81 NAPRT (0.60) RAB9ASMN1; SMN2NAPRTKMT2ANPC1
SCHEMBL13360508 0.81 NAPRT (0.60) RAB9ASMN1; SMN2NAPRTKMT2ANPC1
SCHEMBL931481 0.81 NAPRT (0.60) RAB9ASMN1; SMN2NAPRTKMT2ANPC1
SCHEMBL2981251 0.81 NAPRT (0.60) RAB9ASMN1; SMN2NAPRTKMT2ANPC1
SCHEMBL931076 0.80 TDP1 (0.61) RAB9ASMN1; SMN2NAPRTKMT2ANPC1
SCHEMBL13527490 0.80 RAB9A (0.56) RAB9ASMN1; SMN2NAPRTKMT2ANPC1
SCHEMBL3531806 0.80 GAA (0.61) RAB9ASMN1; SMN2NAPRTKMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 206 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6844366-B2 Sulfonamide hydroxamates SYNTEX (U.S.A.) LLC (US) 2005-01-18 US claimed
US-20260070902-A1 SULFONYL DERIVATIVES AS CCR6 INHIBITORS HOFFMANN-LA ROCHE INC. (US) 2026-03-12 US disclosed
EP-4630402-A1 SULFONYL DERIVATIVES AS CCR6 INHIBITORS F. Hoffmann-La Roche AG (CH) 2025-10-15 EP disclosed
US-20250282729-A1 CHEMICAL COMPOUND MANUFACTURE, NEW SALT FORM, AND THERAPEUTIC USES THEREOF EUSTRALIS PHARMACEUTICALS LIMITED (TRADING AS PRESSURA NEURO) (AU) 2025-09-11 US disclosed
US-12351557-B2 Chemical compound manufacture, new salt form, and therapeutic uses thereof EUSTRALIS PHARMACEUTICALS LIMITED (AU) 2025-07-08 US disclosed
US-20240425478-A1 CYCLOPENTYLPYRAZOLE CDK2 INHIBITORS GENENTECH INC (US) 2024-12-26 US disclosed
EP-4448514-A1 TYK2 INHIBITORS AND COMPOSITIONS AND METHODS THEREOF Lynk Pharmaceuticals Co. Ltd. (CN) 2024-10-23 EP disclosed
CN-118401516-A TYK2 inhibitors, compositions and methods thereof 凌科药业(杭州)有限公司 2024-07-26 CN disclosed
WO-2024121013-A1 SULFONYL DERIVATIVES AS CCR6 INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2024-06-13 WO disclosed
US-20240174662-A1 SMALL MOLECULE INHIBITORS OF SALT INDUCIBLE KINASES CILAG AG (CH) 2024-05-30 US disclosed
US-6297375-B1 4-phenyl-pyridine derivatives HOFFMANN-LA ROCHE INC. 2001-10-02 US disclosed
CN-1297887-A Process for producing pyridine derivate HOFFMANN LA ROCHE (CH) 2001-06-06 CN disclosed
EP-1103546-A1 Process for preparation of pyridine derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-05-30 EP disclosed
CN-1270959-A 4-phenyl pyridine derivatives HOFFMANN LA ROCHE (CH) 2000-10-25 CN disclosed
EP-1035115-A1 4-Phenylpyridine derivatives and their use as NK-1 receptor antagonists F. HOFFMANN-LA ROCHE AG (CH) 2000-09-13 EP disclosed
US-4410530-A CARDIO-SELECTIVE B-RECEPTOR BLOCKING AGENTS AND STIMULANTS CIBA-GEIGY CORPORATION (US) 1983-10-18 US disclosed
US-4195090-A ADRENERGIC BLOCKING AGENTS CIBA-GEIGY CORPORATION (US) 1980-03-25 US disclosed
US-4139623-A HYPOTENSIVE AGENTS C-G CORP. (US) 1979-02-13 US disclosed
US-4115575-A CARDIOVASCULAR DISORDERS CIBA-GEIGY CORPORATION (US) 1978-09-19 US disclosed
US-4027027-A BETA-RECEPTOR-BLOCKERS, HYPOTENSIVES AND VALODILATORS; FOR TREATING ARRYTHMIAS AND ANGINA PECTORIS CIBA-GEIGY CORPORATION (US) 1977-05-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240425478-A1 CYCLOPENTYLPYRAZOLE CDK2 INHIBITORS CDK2, CCNI, CDK20 RAB9A 2194/4885SMN1; SMN2 1757/4885NAPRT 1290/4885
US-20260070902-A1 SULFONYL DERIVATIVES AS CCR6 INHIBITORS CCR6, CCR1, CCR4 RAB9A 2194/4885SMN1; SMN2 1277/4885NAPRT 2185/4885
US-20250282729-A1 CHEMICAL COMPOUND MANUFACTURE, NEW SALT FORM, AND THERAPEUTIC USES THEREOF SCN5A, MGMT, NISCH RAB9A 1880/4885SMN1; SMN2 2692/4885NAPRT 2078/4885
US-20240174662-A1 SMALL MOLECULE INHIBITORS OF SALT INDUCIBLE KINASES SIK2, SIK1, SGK2 RAB9A 1869/4885SMN1; SMN2 3406/4885NAPRT 2582/4885
US-12351557-B2 Chemical compound manufacture, new salt form, and therapeutic uses thereof SCN5A, MGMT, NISCH RAB9A 1880/4885SMN1; SMN2 2692/4885NAPRT 2078/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.