SCHEMBL10317092

SCHEMBL10317092

CC(C)(C)OC(=O)NCCNc1cnc(-n2ccc3cc(N(CC(=O)O)S(=O)(=O)c4cc(Cl)cc(Cl)c4)ccc32)cn1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IRAK4 Q9NWZ3 1/20 0.33
SUV39H2 Q9H5I1 3/20 0.32
STK17B O94768 1/20 0.31
STK17A Q9UEE5 1/20 0.31
CKS1B P61024 1/20 0.31
SKP1 P63208 1/20 0.31
SKP2 Q13309 1/20 0.31
BRD4 O60885 2/20 0.31
KEAP1 Q14145 5/20 0.31
NFE2L2 Q16236 5/20 0.31
GNRHR P30968 1/20 0.30
LATS1 O95835 1/20 0.30
CDK2 P24941 1/20 0.30
F2 P00734 1/20 0.30
ALDH1A1 P00352 1/20 0.30
TP53 P04637 1/20 0.30
GLA P06280 1/20 0.30
MAPT P10636 1/20 0.30
HPGD P15428 1/20 0.30
XBP1 P17861 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13390372 0.95 IRAK4 (0.34) IRAK4SUV39H2STK17BSTK17ACKS1B
SCHEMBL3300747 0.90 MAPT (0.33) IRAK4KEAP1NFE2L2F2TP53
SCHEMBL13390518 0.88 CCR9 (0.34) IRAK4TP53MAPTHSD17B10DGAT1
SCHEMBL3301519 0.88 KEAP1 (0.33) IRAK4KEAP1NFE2L2F2ALDH1A1
SCHEMBL3295593 0.87 IRAK4 (0.34) IRAK4SUV39H2STK17BSTK17ACKS1B
SCHEMBL3298992 0.87 KDM4D (0.34) IRAK4KEAP1NFE2L2F2
SCHEMBL3295567 0.86 TMEM97 (0.33) IRAK4KEAP1NFE2L2F2MAPT
SCHEMBL13391255 0.86 PLAU (0.33) IRAK4KEAP1NFE2L2F2ALDH1A1
SCHEMBL13390343 0.86 IRAK4 (0.33) IRAK4TP53MAPTHSD17B10DGAT1
Hydrochloric Acid SCHEMBL3300119 0.86 KEAP1 (0.34) IRAK4KEAP1NFE2L2F2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2121600-B1 SUBSTITUTED ARYLSULPHONYLGLYCINES, THE PREPARATION THEREOF AND THE USE THEREOF AS PHARMACEUTICAL COMPOSITIONS BOEHRINGER INGELHEIM INT (DE) 2012-07-18 EP disclosed