Ziprasidone

Ziprasidone

SCHEMBL10324884

Cl.O.O.O.O=C1Cc2cc(CCN3CCN(c4nsc5ccccc45)CC3)c(Cl)cc2N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

DRD2HTR2AHTR2C

The experimentally established mechanism targets of Ziprasidone. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A known ✓ P28223 13/20 0.96
DRD2 known ✓ P14416 11/20 0.96
HTR2C known ✓ P28335 1/20 0.96
KCNH2 Q12809 2/20 1.00
MTOR P42345 1/20 1.00
RAB9A P51151 1/20 1.00
HTR1A P08908 8/20 0.96
HTR7 P34969 3/20 0.96
HTR6 P50406 2/20 0.96
HTR3E A5X5Y0 1/20 0.96
HTR3B O95264 1/20 0.96
ABCB11 O95342 1/20 0.96
PGR P06401 1/20 0.96
CHRM2 P08172 1/20 0.96
ADRA2A P08913 1/20 0.96
ADORA3 P0DMS8 1/20 0.96
MAPT P10636 1/20 0.96
CHRM1 P11229 1/20 0.96
GOT1 P17174 1/20 0.96
ADRA2B P18089 1/20 0.96

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Ziprasidone SCHEMBL930539 1.00 KCNH2 (1.00) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL1164202 1.00 KCNH2 (1.00) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL122875 1.00 KCNH2 (1.00) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL29594402 1.00 KCNH2 (1.00) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL6061373 1.00 KCNH2 (1.00) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL2978306 1.00 KCNH2 (1.00) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL2978308 1.00 KCNH2 (1.00) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL4914143 0.99 HTR2A (0.98) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL30354044 0.99 HTR2A (0.98) KCNH2MTORRAB9AHTR2ADRD2
Ziprasidone SCHEMBL374870 0.99 HTR2A (0.98) KCNH2MTORRAB9AHTR2ADRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012096632-A1 NEW ADDITION SALTS OF ZIPRASIDONE, A PROCESS FOR THE PREPARATION THEREOF AND USE THEREOF IN THERAPY SILVERSTONE PHARMA AG (LI) 2012-07-19 WO disclosed