SCHEMBL10328512

SCHEMBL10328512

COc1cc2nccc(Cc3ccc(NS(=O)(=O)c4ccccc4C(F)(F)F)c(C)c3)c2cc1OC

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
AXL P30530 19/20 0.63
SLC22A12 Q96S37 1/20 0.48
EGFR P00533 1/20 0.47
MET P08581 1/20 0.47
SRC P12931 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10328507 0.92 AXL (0.71) AXLEGFRMETSRC
SCHEMBL10328528 0.86 AXL (0.51) AXL
SCHEMBL10328530 0.84 AXL (0.73) AXLEGFRMETSRC
SCHEMBL1590961 0.83 AXL (0.87) AXL
SCHEMBL10328533 0.83 AXL (0.62) AXLEGFRMETSRC
SCHEMBL13667277 0.82 AXL (0.51) AXL
SCHEMBL13667521 0.81 AXL (0.61) AXL
SCHEMBL10328505 0.80 AXL (0.73) AXLEGFRMETSRC
SCHEMBL10328503 0.79 AXL (0.59) AXL
SCHEMBL13667523 0.79 AXL (0.59) AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP disclosed
WO-2009127417-A1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2009-10-22 WO disclosed