SCHEMBL10328528

SCHEMBL10328528

COc1cc2nccc(Cc3ccc(NS(=O)(=O)c4ccc(OC)c5ccccc45)c(C)c3)c2cc1OC

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
AXL P30530 7/20 0.51
FABP4 P15090 5/20 0.48
SMN1; SMN2 Q16637 3/20 0.46
ALDH1A1 P00352 3/20 0.46
KDM4E B2RXH2 1/20 0.46
GAA P10253 1/20 0.46
LMNA P02545 2/20 0.45
HPGD P15428 1/20 0.45
MAPK1 P28482 1/20 0.45
HTT P42858 2/20 0.44
PDE10A Q9Y233 1/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
TSHR P16473 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10328506 0.90 AXL (0.57) AXLFABP4ALDH1A1LMNAHTT
SCHEMBL10328512 0.86 AXL (0.63) AXL
SCHEMBL13667277 0.85 AXL (0.51) AXLSMN1; SMN2GAAMAPK1HTT
SCHEMBL10328533 0.84 AXL (0.62) AXL
SCHEMBL10328508 0.82 AXL (0.44) AXLPDE10AMEN1KMT2A
SCHEMBL1592121 0.81 AXL (0.70) AXL
SCHEMBL10328479 0.81 AXL (0.58) AXLFABP4
SCHEMBL13667521 0.81 AXL (0.61) AXL
SCHEMBL10328489 0.80 AXL (0.58) AXLSMN1; SMN2GAA
SCHEMBL10328503 0.79 AXL (0.59) AXL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2262772-B1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX PLANCK GESELLSCHAFT (DE) 2012-07-18 EP disclosed
WO-2009127417-A1 QUINOLINE DERIVATIVES AS AXL KINASE INHIBITORS MAX-PLANCK-Gesellschaft zur Förderung der Wissenschaften e.V. (DE) 2009-10-22 WO disclosed