SCHEMBL10333296

SCHEMBL10333296

OC(Cc1ccc(C(F)(F)F)cc1)Cn1cncn1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
POLB P06746 1/20 0.41
HPGD P15428 1/20 0.41
HDAC1 Q13547 2/20 0.41
HDAC6 Q9UBN7 2/20 0.41
KMT2A Q03164 2/20 0.39
HSP90AA1 P07900 1/20 0.38
MEN1 O00255 1/20 0.37
KDM4E B2RXH2 1/20 0.37
ALOX15 P16050 1/20 0.37
CYP19A1 P11511 2/20 0.36
CYP3A4 P08684 1/20 0.36
MCHR1 Q99705 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
DNM1 Q05193 1/20 0.36
MC3R P41968 1/20 0.35
PPARG P37231 1/20 0.35
PPARA Q07869 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10333104 0.81 KMT2A (0.51) POLBHPGDHDAC1HDAC6KMT2A
SCHEMBL10333189 0.81 POLB (0.40) POLBHPGDHDAC1HDAC6KMT2A
SCHEMBL11187456 0.80 CYP19A1 (0.41) POLBHPGDHDAC1HDAC6KMT2A
SCHEMBL10333042 0.75 HMOX1 (0.49)
SCHEMBL5925447 0.74 CYP19A1 (0.51) CYP19A1CYP3A4
SCHEMBL14476866 0.74 CYP19A1 (0.56) HDAC1HDAC6CYP19A1
SCHEMBL4249454 0.73 POLB (0.50) POLBHPGDHDAC1HDAC6HSP90AA1
SCHEMBL10333391 0.72 CYP1A2 (0.44) HDAC1HDAC6KMT2AHSP90AA1CYP3A4
SCHEMBL27956483 0.72 HSP90AA1 (0.51) POLBHPGDKMT2AHSP90AA1MEN1
SCHEMBL9826863 0.72 HSP90AA1 (0.54) HDAC1HDAC6KMT2AHSP90AA1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4933357-A 1,3-diazolyl-2-phenylalkyl-2-propanol derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-12 US disclosed
EP-0250198-A2 Bis-azolyl compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-12-23 EP disclosed