SCHEMBL10337607

SCHEMBL10337607

O=C(O)NC1CCN(c2nc3ccccc3n2Cc2ccc(F)cc2)CC1

nearest known ligand 0.74

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HRH1 P35367 18/20 0.74
CYP2D6 P10635 17/20 0.74
CHRM1 P11229 6/20 0.74
KCNH2 Q12809 9/20 0.64
HTR3A P46098 1/20 0.63
CYP3A4 P08684 1/20 0.59
SSTR5 P35346 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15568527 0.87 HRH1 (0.66) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL27317913 0.85 HRH1 (0.69) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL5226378 0.85 HRH1 (1.00) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL31553435 0.85 HRH1 (1.00) HRH1CYP2D6CHRM1KCNH2HTR3A
Water SCHEMBL10337970 0.84 HRH1 (0.98) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL5229655 0.83 HRH1 (0.73) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL11479448 0.83 SSTR5 (0.81) HRH1CYP2D6CHRM1KCNH2HTR3A
Trifluoroacetic Acid SCHEMBL15567418 0.83 HRH1 (0.59) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL15568620 0.82 HRH1 (0.63) HRH1CYP2D6CHRM1KCNH2HTR3A
SCHEMBL10483537 0.82 HRH1 (0.80) HRH1CYP2D6CHRM1KCNH2HTR3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-4912219-A 2-[4-pyrimidin-2-yl amino)piperidin-1-yl]benzimidazole compound SYNTHELABO (FR) 1990-03-27 US disclosed
US-4820710-A ANTIALLERGENS, ANTIHISTAMINES, ANTIINFLAMMATORY AGENTS SYNTHELABO (FR) 1989-04-11 US disclosed