SCHEMBL10345211

SCHEMBL10345211

CN1CCCC(O)(COc2ccccc2)C1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
CYP3A4 P08684 1/20 0.46
TDP1 Q9NUW8 1/20 0.44
DRD2 P14416 1/20 0.40
ALDH1A1 P00352 2/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
KMT2A Q03164 1/20 0.39
SMN1; SMN2 Q16637 2/20 0.38
KDM4E B2RXH2 1/20 0.38
DRD4 P21917 1/20 0.38
OPRM1 P35372 1/20 0.38
CYP1A2 P05177 2/20 0.38
NPC1 O15118 1/20 0.38
POLB P06746 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HPGD P15428 1/20 0.38
CYP2C19 P33261 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL10345286 0.99 TSHR (0.49) TSHRCYP3A4TDP1DRD2ALDH1A1
SCHEMBL10345242 0.79 CYP2D6 (0.55) TSHRCYP3A4ALDH1A1MEN1KMT2A
Hydrochloric Acid SCHEMBL10345025 0.78 CYP2D6 (0.54) TSHRCYP3A4ALDH1A1MEN1KMT2A
SCHEMBL28914522 0.75 ALDH1A1 (0.45) TDP1ALDH1A1MEN1LMNAKMT2A
SCHEMBL10345158 0.72 CYP3A4 (0.50) TSHRCYP3A4ALDH1A1MEN1KMT2A
SCHEMBL18785455 0.71 DPP7 (0.43) TSHRTDP1MEN1KMT2ADRD4
SCHEMBL25599411 0.70 NPC1 (0.42) TDP1DRD2ALDH1A1DRD4OPRM1
SCHEMBL7953412 0.70 CHRNA7 (0.37) TSHRCYP3A4ALDH1A1CYP1A2CYP2D6
SCHEMBL3443283 0.69 HRH3 (0.51) TSHRCYP3A4DRD2ALDH1A1KDM4E
Hydrochloric Acid SCHEMBL10345271 0.69 CHRNA7 (0.37) TSHRCYP3A4ALDH1A1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0152236-B1 ARYLOXYMETHYLPYRROLIDINOLS AND PIPERIDINOLS HAVING ANTIDEPRESSANT, ANTIARHYTHMIC OR HYPOTENSIVE ACTIVITY A.H. ROBINS COMPANY, INCORPORATED (US) 1990-04-18 EP claimed
EP-0152236-A2 Aryloxymethylpyrrolidinols and piperidinols having antidepressant, antiarhythmic or hypotensive activity A.H. ROBINS COMPANY, INCORPORATED (US) 1985-08-21 EP claimed
US-4508724-A Aryloxymethylpyrrolidinols and piperidinols having antidepressant, antiarrhythmic or hypotensive activity A. H. ROBINS COMPANY, INC. (US) 1985-04-02 US claimed