SCHEMBL10347703

SCHEMBL10347703

CC1(C)Oc2cc([N+](=O)[O-])c(Br)cc2C2OC21

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
ALDH1A1 P00352 3/20 0.33
CYP3A4 P08684 1/20 0.33
MAPT P10636 3/20 0.32
MAPK1 P28482 1/20 0.32
CYP2D6 P10635 1/20 0.31
IDO1 P14902 2/20 0.31
KCNH2 Q12809 1/20 0.31
XDH P47989 1/20 0.30
PKM P14618 1/20 0.30
CTSB P07858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6982321 0.84 CYP1A2 (0.55) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL5989140 0.82 ALDH1A1 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL2883779 0.82 ALDH1A1 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL2882585 0.82 ALDH1A1 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL3947551 0.82 ALDH1A1 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL2887116 0.82 ALDH1A1 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL2882586 0.82 ALDH1A1 (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL9742504 0.81 CYP1A2 (0.55) CYP1A2CYP2C9CYP2C19ALDH1A1CYP3A4
SCHEMBL13476208 0.78 MAPT (0.38) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT
SCHEMBL14765557 0.78 KCNH2 (0.42) CYP1A2CYP2C9CYP2C19ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214818-A2 Active compounds BEECHAM GROUP PLC (GB) 1987-03-18 EP claimed
EP-0214818-B1 ACTIVE COMPOUNDS BEECHAM GROUP PLC (GB) 1990-06-20 EP disclosed
US-4782083-A 3,4-dihydro-2H-1-benzopyrans useful as anti-hypertensive agents BEECHAM GROUP P.L.C. (GB) 1988-11-01 US disclosed
EP-0214818-A2 Active compounds BEECHAM GROUP PLC (GB) 1987-03-18 EP disclosed