SCHEMBL10348273

SCHEMBL10348273

CC1(C)Oc2cc([N+](=O)[O-])c(Br)cc2C(O)C1Br

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
KCNH2 Q12809 1/20 0.38
ALDH1A1 P00352 5/20 0.36
CYP2D6 P10635 1/20 0.36
IDO1 P14902 1/20 0.36
TLR3 O15455 1/20 0.35
MAPT P10636 4/20 0.34
MAPK1 P28482 2/20 0.34
GAA P10253 1/20 0.33
PKM P14618 1/20 0.32
CYP3A4 P08684 1/20 0.32
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
AAK1 Q2M2I8 1/20 0.31
L3MBTL1 Q9Y468 1/20 0.31
ABCC9 O60706 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10348274 1.00 CYP1A2 (0.38) CYP1A2CYP2C9CYP2C19KCNH2ALDH1A1
SCHEMBL10348272 1.00 CYP1A2 (0.38) CYP1A2CYP2C9CYP2C19KCNH2ALDH1A1
SCHEMBL9685149 0.86 CYP1A2 (0.52) CYP1A2CYP2C9CYP2C19KCNH2ALDH1A1
SCHEMBL10347884 0.82 CYP1A2 (0.40) CYP1A2CYP2C9CYP2C19KCNH2ALDH1A1
SCHEMBL10347881 0.82 CYP1A2 (0.40) CYP1A2CYP2C9CYP2C19KCNH2ALDH1A1
SCHEMBL10347880 0.82 CYP1A2 (0.40) CYP1A2CYP2C9CYP2C19KCNH2ALDH1A1
SCHEMBL9200696 0.81 KCNH2 (0.40) KCNH2ALDH1A1IDO1TLR3MAPT
SCHEMBL10892807 0.81 KCNH2 (0.48) CYP1A2KCNH2ALDH1A1MAPTGAA
SCHEMBL9684999 0.81 KCNH2 (0.48) CYP1A2KCNH2ALDH1A1MAPTGAA
SCHEMBL10892820 0.81 KCNH2 (0.48) CYP1A2KCNH2ALDH1A1MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0214818-B1 ACTIVE COMPOUNDS BEECHAM GROUP PLC (GB) 1990-06-20 EP disclosed
US-4782083-A 3,4-dihydro-2H-1-benzopyrans useful as anti-hypertensive agents BEECHAM GROUP P.L.C. (GB) 1988-11-01 US disclosed
EP-0214818-A2 Active compounds BEECHAM GROUP PLC (GB) 1987-03-18 EP disclosed