SCHEMBL10358643

SCHEMBL10358643

OCCc1sc(Nc2ccccc2)nc1-c1ccc(Cl)cc1

nearest known ligand 0.72

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PTGDR2 Q9Y5Y4 16/20 0.72
GAA P10253 4/20 0.72
MAPT P10636 4/20 0.72
MEN1 O00255 4/20 0.72
KMT2A Q03164 4/20 0.72
ALDH1A1 P00352 2/20 0.72
POLB P06746 2/20 0.72
KDM4E B2RXH2 1/20 0.72
SMN1; SMN2 Q16637 1/20 0.57
LMNA P02545 1/20 0.50
ALOX12 P18054 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
DHODH Q02127 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11852874 0.84 PTGDR2 (1.00) PTGDR2GAAMAPTMEN1KMT2A
SCHEMBL14433253 0.82 PTGDR2 (0.65) PTGDR2GAAMAPTMEN1KMT2A
SCHEMBL10358559 0.81 MYC (0.51) PTGDR2GAAMAPTMEN1KMT2A
Carbamic Acid SCHEMBL10359033 0.80 PTGDR2 (0.53) PTGDR2GAAMAPTMEN1KMT2A
SCHEMBL29044444 0.75 GAA (0.59) PTGDR2GAAMAPTMEN1KMT2A
SCHEMBL1884723 0.75 PTGDR2 (0.61) PTGDR2GAAMAPTMEN1KMT2A
Carbamic Acid SCHEMBL10358650 0.74 HTT (0.64) PTGDR2GAAMAPTMEN1KMT2A
SCHEMBL10358535 0.74 HTT (0.73) PTGDR2GAAMAPTMEN1KMT2A
SCHEMBL28250062 0.74 PTGDR2 (0.68) PTGDR2GAAMAPTMEN1KMT2A
SCHEMBL28925053 0.73 PTGDR2 (0.65) PTGDR2GAAMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0267986-B1 \"(2-AMINO-4-ARYL-THIAZOLE-5-YL)ETHANOLS AND THEIR DERIVATIVES HAVING DIURETIC ACTIVITY AND METHODS FOR PREPARING THE SAME ISTITUTO LUSO FARMACO D'ITALIA S.p.A. (IT) 1990-11-22 EP disclosed
US-4761422-A (2-amino-4-aryl-thiazole-5-yl)ethanols and their derivatives having diuretic activity and methods for preparing the same LUSOFARMACO ISTITUTO LUSOFARMACO D'ITALIA SPA (IT) 1988-08-02 US disclosed
EP-0267986-A1 \"(2-amino-4-aryl-thiazole-5-yl)ethanols and their derivatives having diuretic activity and methods for preparing the same ISTITUTO LUSO FARMACO D'ITALIA S.p.A. (IT) 1988-05-25 EP disclosed