SCHEMBL10360757

SCHEMBL10360757

CC(c1c[nH]nn1)C(O)(c1ccc(C(F)(F)F)cc1)c1ccc(C(F)(F)F)cc1

nearest known ligand 0.34

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 3/20 0.34
CYP3A5 P20815 1/20 0.34
TRPV6 Q9H1D0 2/20 0.33
ORAI1 Q96D31 1/20 0.33
ORAI2 Q96SN7 1/20 0.33
ORAI3 Q9BRQ5 1/20 0.33
MGLL Q99685 1/20 0.33
NR1H2 P55055 2/20 0.33
NR1H3 Q13133 2/20 0.33
AHR P35869 1/20 0.31
CYP17A1 P05093 1/20 0.31
CA1 P00915 1/20 0.31
CA2 P00918 1/20 0.31
NOS1 P29475 1/20 0.31
PDE2A O00408 4/20 0.30
KDM4E B2RXH2 1/20 0.30
POLB P06746 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10984883 0.86 CCR6 (0.35) CYP3A4CYP17A1PDE2APOLB
SCHEMBL10872634 0.84 CA1 (0.32) CYP3A4CYP3A5TRPV6ORAI1ORAI2
SCHEMBL10361168 0.81 KDM4E (0.32) CYP3A4CYP3A5CA1CA2KDM4E
SCHEMBL10872520 0.73 CYP19A1 (0.33) CYP3A4CYP17A1
SCHEMBL10980353 0.73 CYP19A1 (0.42) CYP3A4CYP3A5CYP17A1KDM4E
SCHEMBL10360755 0.70 CYP3A4 (0.34) CYP3A4CYP3A5AHRCYP17A1PDE2A
SCHEMBL11221170 0.69
SCHEMBL4953035 0.68
SCHEMBL11141011 0.68 CASR (0.38) CYP3A4CYP17A1
SCHEMBL10872968 0.68 CYP19A1 (0.34) CYP3A4CYP17A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0158448-A2 Azolyl propanols IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-10-16 EP claimed
EP-0158448-B1 AZOLYL PROPANOLS IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-08-29 EP disclosed
US-4833159-A FUNGICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1989-05-23 US disclosed
US-4689337-A 1,2,4-TRIAZOLYL AND PYRAZOLYL GROUPS; FUNGICIDES IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1987-08-25 US disclosed
EP-0158448-A2 Azolyl propanols IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1985-10-16 EP disclosed