SCHEMBL1036396

SCHEMBL1036396

Cc1ncsc1CCOc1cccc(C=C2CCN(C(=O)Nc3cnoc3)CC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 4/20 0.45
CYP2D6 P10635 4/20 0.45
OGA O60502 6/20 0.41
FAAH O00519 4/20 0.39
GABRA1 P14867 1/20 0.39
ADRA2C P18825 1/20 0.39
CNR1 P21554 1/20 0.39
HTR2A P28223 1/20 0.39
HTR2C P28335 1/20 0.39
CNR2 P34972 1/20 0.39
HTR2B P41595 1/20 0.39
TMEM97 Q5BJF2 1/20 0.39
SIGMAR1 Q99720 1/20 0.39
HPGD P15428 3/20 0.38
GAA P10253 1/20 0.35
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1075972 0.86 CYP3A4 (0.42) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1038304 0.86 CYP3A4 (0.49) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1033392 0.85 CYP3A4 (0.46) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1033159 0.85 CYP2D6 (0.48) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1037459 0.84 CYP3A4 (0.41) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1036480 0.84 OGA (0.47) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1037523 0.83 CYP3A4 (0.48) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1033874 0.83 CYP3A4 (0.46) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1035719 0.83 CYP3A4 (0.47) CYP3A4CYP2D6OGAFAAHGABRA1
SCHEMBL1082548 0.83 FAAH (0.56) CYP3A4CYP2D6OGAFAAHGABRA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2276738-A1 ETHER BENZYLIDENE PIPERIDINE 5-MEMBERED ARYL CARBOXAMIDE COMPOUNDS USEFUL AS FAAH INHIBITORS Pfizer Inc. (US) 2011-01-26 EP disclosed
WO-2009127943-A1 ETHER BENZYLIDENE PIPERIDINE 5-MEMBERED ARYL CARBOXAMIDE COMPOUNDS USEFUL AS FAAH INHIBITORS PFIZER INC. (US) 2009-10-22 WO disclosed