SCHEMBL10366754

SCHEMBL10366754

COc1ccc2cc(-c3cc(C)cs3)ccc2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNFRSF1A P19438 3/20 0.40
ADORA1 P30542 1/20 0.38
ABL1 P00519 1/20 0.38
HPGD P15428 1/20 0.36
NCF1 P14598 1/20 0.36
BACE1 P56817 3/20 0.35
GABRA1 P14867 1/20 0.35
GABRG2 P18507 1/20 0.35
GABRB3 P28472 1/20 0.35
GABRA5 P31644 1/20 0.35
GABRA3 P34903 1/20 0.35
GABRA2 P47869 1/20 0.35
NCK1 P16333 1/20 0.35
CTSD P07339 1/20 0.35
HDAC3 O15379 2/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC2 Q92769 2/20 0.34
CHEK1 O14757 1/20 0.34
CLK1 P49759 1/20 0.34
PDGFRB P09619 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10365994 0.79 GABRA1 (0.34) TNFRSF1AGABRA1GABRG2GABRB3GABRA5
SCHEMBL16573997 0.79 PDGFRB (0.46) ADORA1HPGDBACE1NCK1HDAC2
SCHEMBL28147641 0.78 HDAC1 (0.40) TNFRSF1AABL1BACE1GABRA1GABRG2
SCHEMBL29630926 0.77 CYP2A6 (0.54) PDGFRBPDGFRAPIK3CDPIP5K1CPIK3CA
SCHEMBL11957099 0.74 HDAC1 (0.39) TNFRSF1AABL1BACE1GABRA1GABRG2
SCHEMBL423324 0.74 CYP1A2 (0.59) HPGDNCF1BACE1NCK1
SCHEMBL13183567 0.73 CYP1A2 (0.50) TNFRSF1AABL1HPGDBACE1GABRA1
SCHEMBL12695592 0.72 BACE1 (0.57) ADORA1HPGDBACE1PDGFRBPDGFRA
SCHEMBL13183630 0.72 CYP2A6 (0.52) TNFRSF1AABL1HPGDBACE1NCK1
SCHEMBL15344999 0.71 HPGD (0.46) ADORA1ABL1HPGDPDGFRBPDGFRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0190857-B1 QUINOLONE INOTROPIC AGENTS Pfizer Limited (GB) 1990-03-21 EP disclosed
US-4728654-A CONGESTIVE HEART FAILURE PFIZER INC. (US) 1988-03-01 US disclosed
EP-0190857-A2 Quinolone inotropic agents Pfizer Limited (GB) 1986-08-13 EP disclosed