SCHEMBL10367404

SCHEMBL10367404

CC=CCCc1ccc(-c2ccccc2)s1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 5/20 0.51
CYP2C19 P33261 4/20 0.51
CYP2C9 P11712 3/20 0.51
CYP2E1 P05181 2/20 0.51
CYP3A4 P08684 2/20 0.51
CYP2B6 P20813 2/20 0.51
TRPV1 Q8NER1 5/20 0.45
CYP11B1 P15538 1/20 0.40
CYP11B2 P19099 1/20 0.40
HDAC3 O15379 2/20 0.39
HDAC1 Q13547 2/20 0.39
HDAC2 Q92769 2/20 0.39
HDAC8 Q9BY41 2/20 0.39
NR3C2 P08235 1/20 0.39
HTR6 P50406 1/20 0.36
ME2 P23368 1/20 0.36
ME1 P48163 1/20 0.36
ME3 Q16798 1/20 0.36
HSD17B1 P14061 1/20 0.36
HSD17B2 P37059 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13680908 0.79 CYP2A6 (0.55) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL24040189 0.77 CYP2A6 (0.60) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL10369289 0.76 CYP2A6 (0.47) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL10367268 0.73 CYP2A6 (0.51) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL10961977 0.73 CYP2A6 (0.51) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL7451222 0.73 CYP2A6 (0.51) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL5728736 0.73 CYP2A6 (0.71) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL27968489 0.73 CYP2A6 (0.60) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL11624972 0.73 CYP2A6 (0.60) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4
SCHEMBL4619799 0.72 RPS6KB2 (0.60) CYP2A6CYP2C19CYP2C9CYP2E1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0164075-B1 7-OXABICYCLOHEPTANE SUBSTITUTED THIO PROSTAGLANDIN ANALOGS E.R. Squibb & Sons, Inc. (US) 1990-09-12 EP disclosed