SCHEMBL13680908

SCHEMBL13680908

O=CCCc1ccc(-c2ccccc2)s1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 3/20 0.55
CYP2E1 P05181 2/20 0.55
CYP2C9 P11712 2/20 0.55
CYP2B6 P20813 2/20 0.55
CYP2C19 P33261 2/20 0.55
CYP3A4 P08684 1/20 0.55
TRPV1 Q8NER1 4/20 0.47
CYP11B1 P15538 1/20 0.42
CYP11B2 P19099 1/20 0.42
HDAC1 Q13547 3/20 0.42
HDAC3 O15379 2/20 0.42
HDAC2 Q92769 2/20 0.42
HDAC8 Q9BY41 2/20 0.42
HTR6 P50406 1/20 0.41
NR3C2 P08235 1/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 1/20 0.40
POLB P06746 1/20 0.40
KMT2A Q03164 1/20 0.40
CYP2D6 P10635 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10367404 0.79 CYP2A6 (0.51) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL13680909 0.77 KDM4E (0.55) HDAC1HDAC3HDAC2HDAC8RAB9A
SCHEMBL7451222 0.76 CYP2A6 (0.51) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL10961977 0.76 CYP2A6 (0.51) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL24040189 0.76 CYP2A6 (0.60) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL11624972 0.76 CYP2A6 (0.60) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL5728736 0.76 CYP2A6 (0.71) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL27968489 0.76 CYP2A6 (0.60) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL4619799 0.75 RPS6KB2 (0.60) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19
SCHEMBL17203114 0.72 TRPV1 (0.66) CYP2A6CYP2E1CYP2C9CYP2B6CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed
US-7582658-B2 Bicyclic compound ASAHI KASEI PHARMA CORPORATION (JP) 2009-09-01 US disclosed