SCHEMBL10368024

SCHEMBL10368024

O=c1cc2c(nn1-c1ccc(Cl)cc1)-c1cc(Cl)ccc1CC2

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.50
LMNA P02545 4/20 0.50
HPGD P15428 1/20 0.50
ALOX12 P18054 1/20 0.50
MAPT P10636 8/20 0.46
HTT P42858 3/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
KDM4E B2RXH2 3/20 0.44
KMT2A Q03164 5/20 0.44
MEN1 O00255 4/20 0.44
GAA P10253 2/20 0.44
POLB P06746 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
AOC3 Q16853 2/20 0.42
NPSR1 Q6W5P4 2/20 0.41
F7 P08709 1/20 0.40
PARP1 P09874 1/20 0.40
F3 P13726 1/20 0.40
PARP10 Q53GL7 1/20 0.40
PTGS2 P35354 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10367575 0.92 ALDH1A1 (0.48) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL10367897 0.92 ALDH1A1 (0.48) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL10365972 0.92 ALDH1A1 (0.51) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL10366113 0.90 ALDH1A1 (0.46) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL10365902 0.90 ALDH1A1 (0.46) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL10366668 0.89 ALDH1A1 (0.50) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL10365965 0.88 POLB (0.43) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL10368021 0.88 ALDH1A1 (0.65) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL8130580 0.84 ALDH1A1 (0.46) ALDH1A1LMNAHPGDALOX12MAPT
SCHEMBL7286458 0.82 VHL (0.50) ALDH1A1LMNAHPGDALOX12MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0190367-B1 BENZO ADH BDCINNOLINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND MECIDINAL COMPOSITION CONTAINING THEM Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1990-01-17 EP disclosed
US-4782057-A ANTIDOTES FOR OVERSEDATION, ANXIOLYTICS YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1988-11-01 US disclosed
EP-0190367-A1 BENZO ADh BDCINNOLINE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND MECIDINAL COMPOSITION CONTAINING THEM Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1986-08-13 EP disclosed