SCHEMBL10368231

SCHEMBL10368231

Clc1ccc(C(c2ccc(Cl)cc2)(c2ccns2)n2ccnc2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 13/20 0.64
CYP11B1 P15538 1/20 0.47
CYP11B2 P19099 1/20 0.47
NR1I2 O75469 2/20 0.46
ADORA3 P0DMS8 2/20 0.46
TBXA2R P21731 2/20 0.46
CCKBR P32239 2/20 0.46
OPRK1 P41145 2/20 0.46
SLC6A3 Q01959 2/20 0.46
KCNH2 Q12809 2/20 0.46
NR1H4 Q96RI1 2/20 0.46
MEN1 O00255 1/20 0.46
SLC22A1 O15245 1/20 0.46
KCNN4 O15554 1/20 0.46
GMNN O75496 1/20 0.46
USP2 O75604 1/20 0.46
TRPM2 O94759 1/20 0.46
ABCB11 O95342 1/20 0.46
EGFR P00533 1/20 0.46
CA2 P00918 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10369498 0.85 CYP11B1 (0.68) CYP19A1CYP11B1CYP11B2NR1I2ADORA3
SCHEMBL331966 0.83 CYP19A1 (0.90) CYP19A1CYP11B1CYP11B2NR1I2ADORA3
SCHEMBL16160172 0.79 CYP19A1 (0.62) CYP19A1CYP11B1CYP11B2NR1I2ADORA3
SCHEMBL7156136 0.77 CYP11B1 (0.80) CYP19A1CYP11B1CYP11B2NR1I2ADORA3
SCHEMBL10370788 0.76 CYP19A1 (0.38) CYP19A1TSHRKMT2A
SCHEMBL10508410 0.72 CYP19A1 (0.53) CYP19A1MEN1CYP3A4TSHRMAPK1
SCHEMBL7162563 0.71 CYP11B1 (0.69) CYP19A1CYP11B1CYP11B2NR1I2ADORA3
SCHEMBL10370339 0.70 CYP19A1 (0.66) CYP19A1CYP11B1CYP11B2NR1I2ADORA3
SCHEMBL10370638 0.70 CYP19A1 (1.00) CYP19A1CYP11B1CYP11B2NR1I2ADORA3
SCHEMBL10367810 0.69 CYP19A1 (0.61) CYP19A1CYP11B1CYP11B2NR1I2ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0166556-B1 DIARYLDIAZOLYLMETHANES ELI LILLY AND COMPANY (US) 1990-12-05 EP disclosed
US-4735960-A TREATING ESTROGEN-DEPENDENT DISEASES ELI LILLY AND COMPANY (US) 1988-04-05 US disclosed
US-4602025-A TREATMENT OF ESTROGEN DEPENDENT DISEASES ELI LILLY AND COMPANY (US) 1986-07-22 US disclosed
EP-0166556-A1 Diaryldiazolylmethanes ELI LILLY AND COMPANY (US) 1986-01-02 EP disclosed